SCHEMBL8716291

SCHEMBL8716291

Cc1c(C)c2c(c(C)c1NC=O)CC(C)(CSc1nc3ccccc3s1)O2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.42
CYP1A2 P05177 5/20 0.42
CYP3A4 P08684 4/20 0.42
CYP2C19 P33261 4/20 0.42
GAA P10253 3/20 0.42
MAPT P10636 6/20 0.42
POLB P06746 2/20 0.42
APEX1 P27695 1/20 0.42
RECQL P46063 1/20 0.42
HSD17B10 Q99714 2/20 0.41
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
ALOX5 P09917 2/20 0.38
PKM P14618 1/20 0.38
HPGD P15428 1/20 0.38
CYP2D6 P10635 3/20 0.38
LMNA P02545 3/20 0.38
CYP2C9 P11712 1/20 0.38
MAPK1 P28482 1/20 0.38
HIF1A Q16665 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8719962 0.82 ALDH1A1 (0.43) ALDH1A1CYP1A2CYP3A4CYP2C19GAA
SCHEMBL8713478 0.77
SCHEMBL8716780 0.75 ALOX5 (0.32) ALOX5
SCHEMBL9144283 0.72 SMN1; SMN2 (0.34) ALDH1A1CYP1A2CYP3A4CYP2C19MAPT
SCHEMBL8713512 0.71
SCHEMBL8718923 0.70
SCHEMBL6978968 0.70
SCHEMBL25538031 0.66 CYP1A2 (0.61) ALDH1A1CYP1A2CYP3A4CYP2C19MAPT
SCHEMBL13768047 0.61 CYP1A2 (0.67) ALDH1A1CYP1A2CYP3A4CYP2C19MAPT
SCHEMBL30824973 0.61 CYP1A2 (0.56) ALDH1A1CYP1A2CYP3A4CYP2C19MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5770772-A 4-FORMYLAMINO-2,3,5-TRIMETHYL-1-(2-METHYL-2-PROPENYLOXY) -BENZENE; ARTERIOSCLEROSIS, BRAIN AND CARDIOVASCULAR DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-06-23 US disclosed
US-5594154-A 5-AMINO-2-BROMOMETHYL-2,4,6,7-TETRAMETHYL-2,3-DIHYDROBENZO(B) FURANS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-01-14 US disclosed
US-5478844-A Method of using aminocoumaran derivatives for treating cerebrovascular diseases TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-12-26 US disclosed
EP-0483772-B1 Aminocoumaran derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-09-13 EP disclosed
US-5376681-A Aminocoumaran derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-12-27 US disclosed
EP-0483772-A1 Aminocoumaran derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-05-06 EP disclosed