SCHEMBL8716674

SCHEMBL8716674

Cc1cc(C)cc(N(CCN2CCC(C(=O)c3ccc(F)cc3)CC2)C(=O)c2ccc(N)cc2)c1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.51
HTR2C P28335 3/20 0.51
HTR7 P34969 3/20 0.51
HTR6 P50406 3/20 0.51
ALDH1A1 P00352 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
KDM4E B2RXH2 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
HSD11B1 P28845 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8710887 0.93 HSD11B1 (0.51) HTR2AHTR2CHTR7HTR6KDM4E
SCHEMBL8714782 0.92 OPRM1 (0.53) HTR2AHTR2CHTR7HTR6ALDH1A1
SCHEMBL8710989 0.91 HTR2A (0.56) HTR2AHTR2CHTR7HTR6KDM4E
SCHEMBL8714758 0.90 HTR2A (0.48) HTR2AHTR2CHTR7HTR6ALDH1A1
SCHEMBL8710869 0.88 ACHE (0.56) HTR2AHTR2CHTR7HTR6KDM4E
SCHEMBL8711303 0.88 SMN1; SMN2 (0.56) HTR2AHTR2CHTR7HTR6ALDH1A1
SCHEMBL8712288 0.88 HSD11B1 (0.53) HTR2AHTR2CHTR7HTR6ALDH1A1
Fumaric Acid SCHEMBL9232882 0.88 HSD11B1 (0.46) HTR2AHTR2CHTR7HTR6KDM4E
Fumaric Acid SCHEMBL9232880 0.88 HSD11B1 (0.46) HTR2AHTR2CHTR7HTR6KDM4E
SCHEMBL8715993 0.87 HTR2A (0.50) HTR2AHTR2CHTR7HTR6KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5728835-A HYPOTENSIVE AGENTS; ANTIISCHEMIC AGENTS TOA EIYO, LTD. (JP) 1998-03-17 US disclosed
EP-0661266-A1 Substituted cyclic amine compounds as 5HT2 antagonists TOA EIYO LTD. (JP) 1995-07-05 EP disclosed