SCHEMBL8717218

SCHEMBL8717218

NC(=O)c1cccc(C[CH]c2ccccc2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.47
POLB P06746 1/20 0.47
CYP3A4 P08684 1/20 0.47
MAPT P10636 1/20 0.47
TSHR P16473 1/20 0.47
CYP2C19 P33261 1/20 0.47
RECQL P46063 1/20 0.47
BLM P54132 1/20 0.47
PMP22 Q01453 1/20 0.47
HSD17B10 Q99714 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
PRSS1 P07477 1/20 0.46
PRSS2 P07478 1/20 0.46
PRSS3 P35030 1/20 0.46
PLA2G10 O15496 2/20 0.46
PLA2G2A P14555 1/20 0.46
KDM1A O60341 1/20 0.46
MAOA P21397 1/20 0.46
MAOB P27338 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4987201 0.81 MRGPRX4 (0.43) PARP1POLBCYP3A4MAPTTSHR
SCHEMBL8710710 0.80 LOXL2 (0.59) MAPTTSHRFOLH1
SCHEMBL8668550 0.80 UNG (0.62) FOLH1MEP1BUNG
SCHEMBL7785229 0.78 PARP1 (0.44) PARP1POLBCYP3A4MAPTTSHR
SCHEMBL28233593 0.78 PARP1 (0.48) PARP1POLBCYP3A4MAPTTSHR
SCHEMBL4224616 0.78 PLA2G2A (0.69) PARP1POLBCYP3A4MAPTTSHR
SCHEMBL10189495 0.78 PARP1 (0.56) PARP1POLBCYP3A4MAPTTSHR
SCHEMBL27570899 0.77 PARP1 (0.50) PARP1PRSS1PRSS2PRSS3KDM1A
SCHEMBL5881143 0.75 PARP1 (0.53) PARP1POLBCYP3A4MAPTTSHR
SCHEMBL17672270 0.75 PLA2G2A (0.59) PARP1POLBCYP3A4MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5763469-A Substituted cyclic ureas and derivatives thereof useful as retroviral protease inhibitors THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1998-06-09 US disclosed