SCHEMBL8717328

SCHEMBL8717328

CN1CCN(c2c(N)cccc2Cl)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.54
DRD3 P35462 1/20 0.54
ADRA2C P18825 4/20 0.53
KDM4E B2RXH2 2/20 0.47
MAPT P10636 2/20 0.47
POLB P06746 1/20 0.47
RAD52 P43351 1/20 0.47
HTR3A P46098 3/20 0.46
HRH4 Q9H3N8 3/20 0.46
HTR3E A5X5Y0 1/20 0.45
HTR3B O95264 1/20 0.45
HTR3D Q70Z44 1/20 0.45
HTR3C Q8WXA8 1/20 0.45
PTPN11 Q06124 1/20 0.44
ADRA2A P08913 1/20 0.43
CYP2D6 P10635 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA1D P25100 1/20 0.43
ADRA1A P35348 1/20 0.43
ADRA1B P35368 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21448015 0.87 DRD2 (0.63) DRD2DRD3ADRA2CKDM4EMAPT
SCHEMBL22662669 0.83 KEAP1 (0.47) KDM4EMAPTPOLBALDH1A1GAA
SCHEMBL5092052 0.81 KEAP1 (0.50) KDM4EPOLBALDH1A1NPSR1
SCHEMBL29931924 0.81 KEAP1 (0.50) KDM4EPOLBALDH1A1NPSR1
SCHEMBL29512667 0.81 ALDH1A1 (0.39) DRD2DRD3ADRA2CHTR3AALDH1A1
Hydrochloric Acid SCHEMBL23043631 0.80 KEAP1 (0.48) KDM4EMAPTPOLBALDH1A1GAA
SCHEMBL21599144 0.80 DRD2 (0.56) DRD2DRD3ADRA2CHTR3AHTR3E
Hydrochloric Acid SCHEMBL29978819 0.80 KEAP1 (0.48) KDM4EMAPTPOLBALDH1A1GAA
SCHEMBL20180553 0.80 DRD2 (0.56) DRD2DRD3ADRA2CKDM4EMAPT
SCHEMBL29512615 0.79 ALDH1A1 (0.44) PTPN11ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998031669-A1 NOVEL ARYLPIPERAZINE DERIVED FROM PIPERIDINE AS ANTIDEPRESSANT MEDICINES PIERRE FABRE MEDICAMENT (FR) 1998-07-23 WO disclosed
WO-1997014689-A1 ARYL-PIPERAZINE CYCLIC AMINE DERIVATIVES, PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME PIERRE FABRE MEDICAMENT (FR) 1997-04-24 WO disclosed