SCHEMBL871785

SCHEMBL871785

O=C(Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3CCCN3C(=O)Cc3ccccc3Oc3ccccc3)cc2)cc1)[C@@H]1CCCN1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 3/20 0.43
HCRTR2 O43614 3/20 0.43
PABPC1 P11940 1/20 0.43
MAPK1 P28482 2/20 0.43
ALDH1A1 P00352 2/20 0.43
HTT P42858 1/20 0.43
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
CFD P00746 2/20 0.42
PFKFB2 O60825 3/20 0.41
PFKFB1 P16118 3/20 0.41
PFKFB3 Q16875 3/20 0.41
NPSR1 Q6W5P4 3/20 0.40
GAA P10253 1/20 0.40
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.40
EP300 Q09472 1/20 0.39
CREBBP Q92793 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845567 0.92 ALDH1A1 (0.50) HCRTR1HCRTR2PABPC1MAPK1ALDH1A1
SCHEMBL872535 0.90 KDM4E (0.46) PABPC1ALDH1A1PFKFB2PFKFB1PFKFB3
SCHEMBL845110 0.86 ALDH1A1 (0.48) HCRTR1HCRTR2ALDH1A1CYP2C9CYP2C19
SCHEMBL873862 0.86 ALDH1A1 (0.45) PABPC1MAPK1ALDH1A1HTTCYP2C9
SCHEMBL845618 0.82 MAPK1 (0.56) PABPC1MAPK1ALDH1A1HTTCYP2C9
SCHEMBL13272387 0.81 HCRTR1 (0.42) HCRTR1HCRTR2PABPC1MAPK1ALDH1A1
SCHEMBL845353 0.81 KDM4E (0.52) PABPC1MAPK1ALDH1A1CYP2C9CYP2C19
SCHEMBL10119687 0.80 CYP2C9 (0.44) PABPC1MAPK1ALDH1A1HTTCYP2C9
SCHEMBL845305 0.80 GAA (0.58) HCRTR1HCRTR2PABPC1MAPK1ALDH1A1
SCHEMBL845279 0.80 ALDH1A1 (0.53) MAPK1ALDH1A1HTTCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed