SCHEMBL873862

SCHEMBL873862

O=C(Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3CCCN3C(=O)c3ccccc3Oc3ccccc3)cc2)cc1)[C@@H]1CCCN1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
MAPK1 P28482 2/20 0.45
HTT P42858 1/20 0.45
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
PABPC1 P11940 1/20 0.43
PFKFB2 O60825 2/20 0.43
PFKFB1 P16118 2/20 0.43
PFKFB3 Q16875 2/20 0.43
NPSR1 Q6W5P4 2/20 0.42
GAA P10253 2/20 0.41
TSHR P16473 2/20 0.41
POLB P06746 1/20 0.41
EP300 Q09472 1/20 0.41
CREBBP Q92793 1/20 0.41
TRPV1 Q8NER1 1/20 0.40
ROCK2 O75116 1/20 0.40
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.40
DPP4 P27487 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845021 0.91 ALDH1A1 (0.53) ALDH1A1MAPK1HTTCYP2C9CYP2C19
SCHEMBL874313 0.91 MAPK1 (0.50) ALDH1A1MAPK1HTTCYP2C9CYP2C19
SCHEMBL873465 0.89 KDM4E (0.47) ALDH1A1PABPC1PFKFB2PFKFB1PFKFB3
SCHEMBL872930 0.88 GAA (0.52) MAPK1CYP2C9CYP2C19PABPC1GAA
SCHEMBL874056 0.86 TRPV1 (0.42) ALDH1A1MAPK1HTTCYP2C9CYP2C19
SCHEMBL871785 0.86 HCRTR1 (0.43) ALDH1A1MAPK1HTTCYP2C9CYP2C19
SCHEMBL10119619 0.85 MAPK1 (0.46) ALDH1A1MAPK1HTTCYP2C9CYP2C19
SCHEMBL10119315 0.84 MAPT (0.40) ALDH1A1MAPK1HTTCYP2C9CYP2C19
SCHEMBL874324 0.84 MAPK1 (0.42) ALDH1A1MAPK1HTTCYP2C9CYP2C19
SCHEMBL872532 0.84 TRPV1 (0.44) ALDH1A1MAPK1HTTCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed