SCHEMBL872535

SCHEMBL872535

O=C(Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3CCCN3C(=O)Cc3ccccc3OCc3ccccc3)cc2)cc1)[C@@H]1CCCN1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.46
LMNA P02545 1/20 0.46
APP P05067 6/20 0.44
HSD17B10 Q99714 1/20 0.43
ALDH1A1 P00352 3/20 0.43
TSHR P16473 2/20 0.43
KDM1A O60341 1/20 0.43
RCOR1 Q9UKL0 1/20 0.43
NPSR1 Q6W5P4 1/20 0.42
HTR2C P28335 1/20 0.42
HTR2B P41595 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
GAA P10253 1/20 0.40
PFKFB2 O60825 1/20 0.40
PFKFB1 P16118 1/20 0.40
PFKFB3 Q16875 1/20 0.40
PABPC1 P11940 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845353 0.92 KDM4E (0.52) KDM4ELMNAAPPHSD17B10ALDH1A1
SCHEMBL871785 0.90 HCRTR1 (0.43) KDM4ELMNAALDH1A1NPSR1GAA
SCHEMBL845110 0.88 ALDH1A1 (0.48) KDM4ELMNAHSD17B10ALDH1A1KDM1A
SCHEMBL873465 0.88 KDM4E (0.47) KDM4ELMNAAPPHSD17B10ALDH1A1
SCHEMBL845305 0.82 GAA (0.58) KDM4ELMNAALDH1A1TSHRL3MBTL1
SCHEMBL845279 0.81 ALDH1A1 (0.53) KDM4ELMNAAPPALDH1A1NPSR1
SCHEMBL845567 0.81 ALDH1A1 (0.50) KDM4ELMNAALDH1A1NPSR1GAA
SCHEMBL845503 0.81 SGMS2 (0.52) KDM4ELMNAAPPHSD17B10ALDH1A1
SCHEMBL871691 0.80 ALDH1A1 (0.44) KDM4ELMNAHSD17B10ALDH1A1TSHR
SCHEMBL845618 0.80 MAPK1 (0.56) LMNAALDH1A1NPSR1GAAPABPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed