SCHEMBL8718028

SCHEMBL8718028

COC(=O)NC1CCc2sc(Cl)c(C(=O)CCC(=O)O)c2C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.35
POLB P06746 1/20 0.35
MTNR1A P48039 5/20 0.33
MTNR1B P49286 5/20 0.33
KDM4E B2RXH2 2/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
ACHE P22303 1/20 0.32
MAPT P10636 3/20 0.32
SMN1; SMN2 Q16637 2/20 0.31
HPGD P15428 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
ALOX15 P16050 1/20 0.31
DUSP3 P51452 1/20 0.31
PTPN5 P54829 1/20 0.31
PTPN11 Q06124 1/20 0.31
LMNA P02545 1/20 0.31
STING1 Q86WV6 1/20 0.31
HTR1A P08908 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8720199 0.76 HTT (0.38) ALDH1A1MTNR1AMTNR1BCA1CA2
SCHEMBL8718069 0.74 ALDH1A1 (0.44) ALDH1A1LMNASTING1
SCHEMBL8719860 0.72 STING1 (0.41) ALDH1A1MTNR1AMTNR1BCA1CA2
SCHEMBL8718584 0.66 NPC1 (0.41) ALDH1A1MTNR1AMTNR1BCA1CA2
SCHEMBL31564105 0.64 BTK (0.40) CA1CA2DRD2
SCHEMBL21597724 0.63 CA1 (0.56) ALDH1A1POLBCA1CA2ACHE
SCHEMBL21597643 0.63 CA1 (0.56) ALDH1A1POLBCA1CA2ACHE
SCHEMBL8718179 0.62 MTNR1A (0.44) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL21597657 0.61 MAPT (0.55) ALDH1A1POLBKDM4EMAPTSMN1; SMN2
SCHEMBL21597712 0.61 KDM4E (0.47) ALDH1A1KDM4EMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739132-A ENDOTHOXIN SHOCK; NEPHRITIS TANABE SEIYAKU CO., LTD. (JP) 1998-04-14 US disclosed
EP-0579059-A1 Pyridazinone derivatives and processes for preparing the same TANABE SEIYAKU CO., LTD. (JP) 1994-01-19 EP disclosed