SCHEMBL8720199

SCHEMBL8720199

COC(=O)NC1CCc2scc(C(=O)CCC(=O)O)c2C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MTNR1A P48039 7/20 0.37
MTNR1B P49286 7/20 0.37
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
ACHE P22303 1/20 0.36
CYP1A2 P05177 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
ALOX15 P16050 1/20 0.36
HTR1A P08908 1/20 0.35
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35
HTR1B P28222 1/20 0.35
HTR1E P28566 1/20 0.35
HTR7 P34969 1/20 0.35
OPRM1 P35372 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8718028 0.76 ALDH1A1 (0.35) ALDH1A1HPGDMTNR1AMTNR1BCA1
SCHEMBL8719860 0.75 STING1 (0.41) ALDH1A1MTNR1AMTNR1BCA1CA2
SCHEMBL8718069 0.75 ALDH1A1 (0.44) ALDH1A1L3MBTL1
SCHEMBL31564412 0.72 PARP1 (0.39) HTTALDH1A1HPGDL3MBTL1DRD2
SCHEMBL31563964 0.71 ALDH1A1 (0.44) HTTALDH1A1HPGDL3MBTL1MAPT
SCHEMBL31563897 0.68 DRD2 (0.40) HTTALDH1A1L3MBTL1MTNR1AMTNR1B
SCHEMBL8718179 0.68 MTNR1A (0.44) MTNR1AMTNR1BCA1CA2ACHE
SCHEMBL31563929 0.68 CTSK (0.40) HTTALDH1A1HPGDL3MBTL1CA1
SCHEMBL31564232 0.68 DRD2 (0.40) L3MBTL1DRD2
SCHEMBL8714966 0.68 MTNR1A (0.33) HTTALDH1A1HPGDL3MBTL1MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739132-A ENDOTHOXIN SHOCK; NEPHRITIS TANABE SEIYAKU CO., LTD. (JP) 1998-04-14 US disclosed
EP-0579059-A1 Pyridazinone derivatives and processes for preparing the same TANABE SEIYAKU CO., LTD. (JP) 1994-01-19 EP disclosed