SCHEMBL8718199

SCHEMBL8718199

CC(=O)NC(C)(NC(C)=O)P(=O)(O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.39
FDPS P14324 1/20 0.38
EPHX1 P07099 1/20 0.34
CA2 P00918 2/20 0.32
MMP2 P08253 2/20 0.32
MMP8 P22894 2/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
MMP1 P03956 1/20 0.32
MMP9 P14780 1/20 0.32
CA9 Q16790 1/20 0.32
KDM4E B2RXH2 1/20 0.32
PTGS1 P23219 1/20 0.32
MMP12 P39900 1/20 0.32
MMP3 P08254 1/20 0.31
PGK1 P00558 1/20 0.31
PGK2 P07205 1/20 0.31
NFKB1 P19838 1/20 0.30
CYP1A2 P05177 1/20 0.30
PKM P14618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11664388 0.81 LMNA (0.41) LMNAFDPSEPHX1CA2MMP2
SCHEMBL8985384 0.79 EPHX1 (0.39) LMNAFDPSEPHX1CA2MMP2
SCHEMBL28305379 0.73 LMNA (0.35) LMNAFDPSEPHX1
SCHEMBL8720991 0.70 HDAC3 (0.43) FDPSCA2MMP2MMP8CA12
SCHEMBL11659802 0.69 PKM (0.34) FDPSCA2MMP2MMP8CA12
Phosphoric Acid SCHEMBL27902534 0.69 KDM4E (0.38) EPHX1KDM4EPKM
SCHEMBL124179 0.67
SCHEMBL27265453 0.67 EPHX1 (0.42) LMNAEPHX1CA2KDM4EPTGS1
SCHEMBL6363154 0.67
SCHEMBL11664344 0.67 LMNA (0.43) LMNAFDPSCA2MMP2MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0570380-B1 NOVEL METHYLENEBISPHOSPHONIC ACID DERIVATIVES LEIRAS OY (FI) 1998-09-16 EP disclosed
US-5442101-A Treatment of calcium metabolism disorders, bone disorders LEIRAS OY (FI) 1995-08-15 US disclosed
EP-0570380-A1 NOVEL METHYLENEBISPHOSPHONIC ACID DERIVATIVES LEIRAS OY (FI) 1993-11-24 EP disclosed
WO-1992011268-A1 NOVEL METHYLENEBISPHOSPHONIC ACID DERIVATIVES LEIRAS OY (FI) 1992-07-09 WO disclosed