SCHEMBL8720245

SCHEMBL8720245

O=C(O)Cc1ccc(C(=O)c2cccc([N+](=O)[O-])c2)cc1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.58
CES2 O00748 1/20 0.55
CES1 P23141 1/20 0.55
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
ALDH1A1 P00352 4/20 0.53
TSHR P16473 2/20 0.53
THRA P10827 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
MAPT P10636 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
SMN1; SMN2 Q16637 2/20 0.50
HPGD P15428 1/20 0.50
ACHE P22303 1/20 0.50
TDP1 Q9NUW8 1/20 0.49
KMO O15229 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11670232 0.85 TSHR (0.59) TP53CES2CES1MEN1KMT2A
SCHEMBL333455 0.85 TP53 (0.73) TP53CES2CES1MEN1KMT2A
SCHEMBL8720282 0.84 MEN1 (0.58) TP53CES2CES1MEN1KMT2A
SCHEMBL11758821 0.83 TP53 (0.77) TP53CES2CES1MEN1KMT2A
Phosphine SCHEMBL28281304 0.83 TP53 (0.71) TP53CES2CES1MEN1KMT2A
SCHEMBL3234327 0.83 CES2 (0.68) TP53CES2CES1MEN1KMT2A
SCHEMBL11295596 0.83 TP53 (0.71) TP53CES2CES1MEN1KMT2A
SCHEMBL27787065 0.83 TP53 (0.71) TP53CES2CES1MEN1KMT2A
Bicarbonate SCHEMBL27282989 0.83 TP53 (0.71) TP53CES2CES1MEN1KMT2A
Ammonia Solution, Strong SCHEMBL27493385 0.83 TP53 (0.71) TP53CES2CES1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998045298-A1 ANTIVIRAL AGENTS SMITHKLINE BEECHAM PLC (GB) 1998-10-15 WO disclosed