SCHEMBL8720486

SCHEMBL8720486

CSc1nc(Oc2cccc(C(F)(F)F)c2)cc(N(C)C)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.46
MEN1 O00255 1/20 0.45
HTT P42858 1/20 0.45
KMT2A Q03164 1/20 0.45
PDGFRB P09619 1/20 0.44
KIT P10721 1/20 0.44
PDGFRA P16234 1/20 0.44
CDK11B P21127 1/20 0.44
FLT3 P36888 1/20 0.44
CDKL2 Q92772 1/20 0.44
BRAF P15056 1/20 0.42
KDR P35968 1/20 0.42
MAPK14 Q16539 1/20 0.42
TNNI3K Q59H18 1/20 0.42
ALDH1A1 P00352 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
POLB P06746 1/20 0.42
MAPK1 P28482 1/20 0.40
KDM4E B2RXH2 2/20 0.39
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8720487 0.86 MEN1 (0.45) MAPTMEN1HTTKMT2APDGFRB
SCHEMBL8667374 0.84 MAPT (0.48) MAPTMEN1HTTKMT2APDGFRB
SCHEMBL8666887 0.82 MAPT (0.47) MAPTMEN1HTTKMT2APDGFRB
SCHEMBL8672947 0.82 MAPT (0.50) MAPTMEN1HTTKMT2APDGFRB
SCHEMBL8664642 0.82 MAPT (0.47) MAPTMEN1HTTKMT2APDGFRB
SCHEMBL8664737 0.81 MAPK1 (0.51) MAPTMEN1HTTKMT2APDGFRB
SCHEMBL8720532 0.80 POLB (0.46) MAPTHTTBRAFKDRMAPK14
SCHEMBL8723510 0.79 MAPT (0.52) MAPTBRAFKDRMAPK14TNNI3K
SCHEMBL8720496 0.79 ALDH1A1 (0.50) MAPTMEN1KMT2ABRAFKDR
SCHEMBL8668427 0.79 GAA (0.51) MAPTMEN1HTTKMT2APDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700391-B1 HERBICIDAL COMPOUNDS SHELL INT RESEARCH (NL) 1998-10-21 EP disclosed
US-5759956-A PYRAZINE CARBOXAMIDE DERIVATIVES AMERICAN CYANAMID COMPANY (US) 1998-06-02 US disclosed
EP-0700391-A1 HERBICIDAL COMPOUNDS SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1996-03-13 EP disclosed
WO-1994027974-A1 HERBICIDAL COMPOUNDS SHELL INTERNATIONALE RESEARCH MAATSCHAPPIJ B.V. (NL) 1994-12-08 WO disclosed