SCHEMBL8720532

SCHEMBL8720532

CN(C)c1cc(Oc2cccc(C(F)(F)F)c2)nc(C#N)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.46
MAPT P10636 2/20 0.45
CYP1A2 P05177 2/20 0.44
CYP2C9 P11712 2/20 0.44
CYP2C19 P33261 2/20 0.44
RECQL P46063 1/20 0.44
CTSK P43235 8/20 0.44
CTSS P25774 3/20 0.44
BRAF P15056 1/20 0.41
KDR P35968 1/20 0.41
MAPK14 Q16539 1/20 0.41
TNNI3K Q59H18 1/20 0.41
L3MBTL1 Q9Y468 3/20 0.41
ALDH1A1 P00352 2/20 0.41
NPSR1 Q6W5P4 1/20 0.40
KCNH2 Q12809 6/20 0.40
MAPK1 P28482 2/20 0.39
CTSL P07711 2/20 0.39
CTSB P07858 2/20 0.39
F10 P00742 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8720537 0.86 CTSK (0.43) MAPTCTSKCTSSBRAFKDR
SCHEMBL8720486 0.80 MAPT (0.46) POLBMAPTCYP1A2CYP2C9CYP2C19
SCHEMBL8720496 0.78 ALDH1A1 (0.50) POLBMAPTBRAFKDRMAPK14
SCHEMBL8723510 0.78 MAPT (0.52) POLBMAPTCYP1A2CYP2C9CYP2C19
SCHEMBL8720576 0.78 MAPT (0.48) POLBMAPTCYP1A2CYP2C9CYP2C19
SCHEMBL8720577 0.77 MAPT (0.51) POLBMAPTCYP1A2CYP2C9CYP2C19
SCHEMBL8773215 0.77 CYP1A2 (0.50) POLBMAPTCYP1A2CYP2C9CYP2C19
SCHEMBL29607569 0.77 MAPT (0.52) POLBMAPTCYP1A2CYP2C9CYP2C19
SCHEMBL7110308 0.74 POLB (0.51) POLBMAPTCYP1A2CYP2C9CYP2C19
SCHEMBL7110336 0.73 MAPT (0.49) POLBMAPTCYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700391-B1 HERBICIDAL COMPOUNDS SHELL INT RESEARCH (NL) 1998-10-21 EP disclosed
US-5759956-A PYRAZINE CARBOXAMIDE DERIVATIVES AMERICAN CYANAMID COMPANY (US) 1998-06-02 US disclosed
EP-0700391-A1 HERBICIDAL COMPOUNDS SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1996-03-13 EP disclosed
WO-1994027974-A1 HERBICIDAL COMPOUNDS SHELL INTERNATIONALE RESEARCH MAATSCHAPPIJ B.V. (NL) 1994-12-08 WO disclosed