SCHEMBL8720537

SCHEMBL8720537

CN(C)c1cc(Oc2ccc(C(F)(F)F)cc2)nc(C#N)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 5/20 0.43
CTSS P25774 4/20 0.43
KDM4E B2RXH2 3/20 0.42
MAPT P10636 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
SCN9A Q15858 1/20 0.41
LMNA P02545 4/20 0.40
BRAF P15056 1/20 0.39
KDR P35968 1/20 0.39
MAPK14 Q16539 1/20 0.39
TNNI3K Q59H18 1/20 0.39
NPSR1 Q6W5P4 2/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
THRB P10828 1/20 0.37
SLC6A4 P31645 1/20 0.36
UCHL1 P09936 1/20 0.36
USP30 Q70CQ3 1/20 0.36
LIPE Q05469 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8720532 0.86 POLB (0.46) CTSKCTSSKDM4EMAPTL3MBTL1
SCHEMBL8720487 0.78 MEN1 (0.45) KDM4EMAPTL3MBTL1LMNABRAF
SCHEMBL8723515 0.76 SLC6A2 (0.43) KDM4EMAPTL3MBTL1SCN9ALMNA
SCHEMBL8722832 0.76 BRAF (0.45) KDM4EMAPTL3MBTL1SCN9ALMNA
SCHEMBL29608122 0.75 KDM4E (0.50) KDM4EMAPTL3MBTL1SCN9ALMNA
SCHEMBL17908 0.74 LMNA (0.42) CTSKCTSSKDM4EMAPTSCN9A
SCHEMBL8720519 0.73 KMT2A (0.36) CTSKMAPTLMNANPSR1ALDH1A1
SCHEMBL4374883 0.69 LMNA (0.42) KDM4EMAPTSCN9ALMNANPSR1
SCHEMBL23221440 0.68 SLC6A2 (0.40) KDM4EMAPTL3MBTL1SCN9ALMNA
SCHEMBL15955567 0.68 AR (0.46) KDM4EMAPTLMNAKDRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700391-B1 HERBICIDAL COMPOUNDS SHELL INT RESEARCH (NL) 1998-10-21 EP disclosed
US-5759956-A PYRAZINE CARBOXAMIDE DERIVATIVES AMERICAN CYANAMID COMPANY (US) 1998-06-02 US disclosed
EP-0700391-A1 HERBICIDAL COMPOUNDS SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1996-03-13 EP disclosed
WO-1994027974-A1 HERBICIDAL COMPOUNDS SHELL INTERNATIONALE RESEARCH MAATSCHAPPIJ B.V. (NL) 1994-12-08 WO disclosed