SCHEMBL8720615

SCHEMBL8720615

CC(C)(C)C(=O)Nc1ncnc2nc[nH]c12

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 9/20 0.58
NPC1 O15118 1/20 0.58
RAB9A P51151 1/20 0.58
BRAF P15056 1/20 0.56
NT5C2 P49902 2/20 0.53
CYP1A2 P05177 1/20 0.52
HIF1A Q16665 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
CREBBP Q92793 1/20 0.52
TP53 P04637 1/20 0.51
TSHR P16473 1/20 0.51
HSD17B10 Q99714 1/20 0.51
NT5E P21589 1/20 0.51
CYP3A4 P08684 1/20 0.50
HTT P42858 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8718918 0.98 BRD4 (0.57) BRD4NPC1RAB9ABRAFNT5C2
SCHEMBL9408577 0.85 BRAF (0.50) BRD4NPC1RAB9ABRAFCYP1A2
SCHEMBL9408571 0.84 BRAF (0.49) BRD4NPC1RAB9ABRAFCYP1A2
SCHEMBL29475418 0.83 BRAF (0.72) BRD4NPC1RAB9ABRAFNT5C2
SCHEMBL536913 0.83 BRAF (0.72) BRD4NPC1RAB9ABRAFNT5C2
SCHEMBL27204265 0.81 BRD4 (0.55) BRD4NPC1RAB9ABRAFNT5C2
SCHEMBL22118772 0.81 BRD4 (0.68) BRD4NPC1RAB9ABRAFNT5C2
SCHEMBL5437612 0.80 BRD4 (0.62) BRD4NPC1RAB9ABRAFNT5C2
SCHEMBL1358803 0.79 SYK (0.46) NPC1RAB9ABRAFHSD17B10
SCHEMBL17362837 0.79 BRD4 (0.58) BRD4NPC1RAB9ABRAFNT5C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5686611-A Nucleoside analogs INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY OF THE ACADEMY OF SCIENCES OF THE CZECH REPUBLIC (CZ) 1997-11-11 US claimed
US-5821357-A REACTING ALPHA-ANOMER ENRICHED 2,2-DIFLUOROCARBOHYDRATE WITH AT LEAST TWO MOLAR EQUIVALENTS OF METAL DERIVATIVE OF NUCLEOBASE IN LOW FREEZING INERT SOLVENT ELI LILLY AND COMPANY (US) 1998-10-13 US disclosed
US-5686611-A Nucleoside analogs INSTITUTE OF ORGANIC CHEMISTRY AND BIOCHEMISTRY OF THE ACADEMY OF SCIENCES OF THE CZECH REPUBLIC (CZ) 1997-11-11 US disclosed
EP-0577303-B1 Stereoselective glycosylation process LILLY CO ELI (US) 1997-10-01 EP disclosed