SCHEMBL8720924

SCHEMBL8720924

BrC1=C(n2ccnc2)CCC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.38
LMNA P02545 3/20 0.36
MAPT P10636 1/20 0.36
ENPP2 Q13822 1/20 0.36
MKNK1 Q9BUB5 1/20 0.36
MKNK2 Q9HBH9 1/20 0.36
NOTUM Q6P988 1/20 0.36
CYP11B2 P19099 3/20 0.36
CYP11B1 P15538 3/20 0.36
CYP2A6 P11509 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
TSHR P16473 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
PDE4A P27815 1/20 0.35
MAPK1 P28482 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8724347 0.86 CYP3A4 (0.45) CYP3A4LMNAMAPTENPP2MKNK1
SCHEMBL8726118 0.80 CYP3A4 (0.45) CYP3A4LMNAMAPTENPP2MKNK1
SCHEMBL8724187 0.73 CYP3A4 (0.35) CYP3A4LMNAMAPTENPP2MKNK1
SCHEMBL29163972 0.73
SCHEMBL8721430 0.72 CYP3A4 (0.34) CYP3A4LMNAMAPTENPP2MKNK1
SCHEMBL8720945 0.72 CYP3A4 (0.38) CYP3A4LMNAMAPTENPP2MKNK1
SCHEMBL8721411 0.70 TSHR (0.51) CYP3A4LMNAMAPTCYP11B2CYP11B1
SCHEMBL8724318 0.69 CYP3A4 (0.33) CYP3A4LMNAMAPTENPP2MKNK1
SCHEMBL8060377 0.67 CYP3A4 (0.43) CYP3A4LMNAMAPTENPP2MKNK1
SCHEMBL8724368 0.67 CYP11B2 (0.44) CYP3A4LMNAMAPTENPP2MKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998000430-A1 IMIDAZOL DERIVATIVES USEFUL AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-01-08 WO disclosed