SCHEMBL8723610

SCHEMBL8723610

N#Cc1cc[c]c(Nc2ccc(F)cc2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 1/20 0.45
TBXA2R P21731 3/20 0.38
KDM4E B2RXH2 3/20 0.37
TP53 P04637 2/20 0.37
DHODH Q02127 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
MAPT P10636 3/20 0.34
ALDH1A1 P00352 2/20 0.33
CTSL P07711 1/20 0.33
CTSB P07858 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
SYK P43405 1/20 0.33
GAA P10253 1/20 0.33
EGFR P00533 2/20 0.33
ERBB2 P04626 1/20 0.33
MAPK10 P53779 1/20 0.33
NPSR1 Q6W5P4 1/20 0.32
MEN1 O00255 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28285324 0.84 CA12 (0.42) KDM4EMAPTALDH1A1GAAEGFR
SCHEMBL8723668 0.79 MAPK10 (0.38) NPC1RAB9AMAPTALDH1A1EGFR
SCHEMBL13352440 0.73 KDM4E (0.52) CDC7TBXA2RKDM4ETP53DHODH
SCHEMBL16481157 0.71 CDC7 (0.71) CDC7KDM4ETP53MAPTALDH1A1
SCHEMBL8725399 0.71 EGFR (0.44) KDM4ENPC1RAB9AMAPTALDH1A1
SCHEMBL27374955 0.69 CDC7 (0.49) CDC7TBXA2RDHODHNPC1RAB9A
SCHEMBL30751294 0.69 CDC7 (0.49) CDC7TBXA2RDHODHNPC1RAB9A
SCHEMBL184366 0.69
SCHEMBL8169486 0.69 PRSS1 (0.39) ALDH1A1
SCHEMBL3932390 0.68 NPC1 (0.41) KDM4EDHODHNPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832091-A1 C-4' MODIFIED ADENOSINE KINASE INHIBITORS GENSIA, INC. (US) 1998-04-01 EP disclosed
WO-1996040705-A1 C-4' MODIFIED ADENOSINE KINASE INHIBITORS GENSIA SICOR (US) 1996-12-19 WO disclosed