SCHEMBL8725399

SCHEMBL8725399

COc1cc[c]c(Nc2ccc(F)cc2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.44
ERBB3 P21860 1/20 0.44
MAOB P27338 2/20 0.41
MAOA P21397 1/20 0.41
MAPK1 P28482 3/20 0.41
MAPT P10636 3/20 0.41
KDM4E B2RXH2 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
NPC1 O15118 1/20 0.41
GAA P10253 1/20 0.41
THRB P10828 1/20 0.41
RECQL P46063 1/20 0.41
RAB9A P51151 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
ALOX15 P16050 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8721645 0.88 MAPT (0.55) MAPK1MAPTKDM4EL3MBTL1NPC1
SCHEMBL28318419 0.83 GAA (0.50) EGFRMAPK1MAPTKDM4EL3MBTL1
SCHEMBL8723668 0.79 MAPK10 (0.38) EGFRMAPK1MAPTNPC1RAB9A
SCHEMBL8721665 0.75 GAA (0.38) EGFRMAPK1MAPTKDM4EL3MBTL1
SCHEMBL4838147 0.73 CA1 (0.35) MAPK1MAPTKDM4EL3MBTL1NPC1
SCHEMBL866356 0.73 MAPT (0.77) EGFRERBB3MAOBMAOAMAPK1
SCHEMBL7844969 0.73 MTNR1B (0.64) MAOBMAPK1MAPTKDM4EL3MBTL1
SCHEMBL8327622 0.71 MAOB (0.43) MAOBMAPTKDM4EL3MBTL1NPC1
SCHEMBL8723610 0.71 CDC7 (0.45) EGFRMAPTKDM4ENPC1GAA
SCHEMBL4242 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832091-A1 C-4' MODIFIED ADENOSINE KINASE INHIBITORS GENSIA, INC. (US) 1998-04-01 EP disclosed
WO-1996040705-A1 C-4' MODIFIED ADENOSINE KINASE INHIBITORS GENSIA SICOR (US) 1996-12-19 WO disclosed