SCHEMBL8723680

SCHEMBL8723680

CN(C)CCNC(=O)c1ccc(Nc2ccccc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.57
HDAC6 Q9UBN7 2/20 0.56
HDAC3 O15379 1/20 0.55
HDAC1 Q13547 1/20 0.55
HDAC2 Q92769 1/20 0.55
HDAC8 Q9BY41 1/20 0.55
AURKA O14965 1/20 0.55
AURKB Q96GD4 1/20 0.55
TDP1 Q9NUW8 1/20 0.53
NAMPT P43490 2/20 0.53
MCHR1 Q99705 1/20 0.53
TMEM97 Q5BJF2 1/20 0.52
SIGMAR1 Q99720 1/20 0.52
ALOX5 P09917 1/20 0.52
IKBKB O14920 1/20 0.52
CHUK O15111 1/20 0.52
IKBKG Q9Y6K9 1/20 0.52
LMNA P02545 1/20 0.51
POLB P06746 1/20 0.51
SETD7 Q8WTS6 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2087431 0.87 ALDH1A1 (0.62) ALDH1A1HDAC6HDAC3HDAC1HDAC2
SCHEMBL1499275 0.87 HDAC1 (0.59) ALDH1A1HDAC6HDAC3HDAC1HDAC2
Hydrochloric Acid SCHEMBL20547794 0.85 ALDH1A1 (0.60) ALDH1A1HDAC6HDAC3HDAC1HDAC2
SCHEMBL1499235 0.85 BRAF (0.56) ALDH1A1AURKAAURKBNAMPTIKBKB
SCHEMBL30046741 0.85 ALDH1A1 (0.73) ALDH1A1HDAC6HDAC3HDAC1HDAC2
SCHEMBL8150809 0.84 NPC1 (0.63) ALDH1A1HDAC6HDAC1MCHR1TMEM97
SCHEMBL12766913 0.84 ALDH1A1 (0.64) ALDH1A1NAMPTSIGMAR1ALOX5POLB
SCHEMBL1499442 0.83 MTNR1B (0.54) ALDH1A1MCHR1ALOX5CYP2D6
SCHEMBL29973388 0.83 MTNR1B (0.54) ALDH1A1MCHR1ALOX5CYP2D6
SCHEMBL5582704 0.83 MCHR1 (0.70) TDP1NAMPTMCHR1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832091-A1 C-4' MODIFIED ADENOSINE KINASE INHIBITORS GENSIA, INC. (US) 1998-04-01 EP disclosed
WO-1996040705-A1 C-4' MODIFIED ADENOSINE KINASE INHIBITORS GENSIA SICOR (US) 1996-12-19 WO disclosed