SCHEMBL8723729

SCHEMBL8723729

O=C(Nc1cc(C2CCC3CCCCN3CC2)c[nH]1)c1ccoc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.42
HTR1D P28221 1/20 0.42
HTR1B P28222 1/20 0.42
HTR1F P30939 1/20 0.42
TMIGD3 P0DMS9 1/20 0.38
ADORA1 P30542 1/20 0.38
KMT2A Q03164 2/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
MAPK14 Q16539 1/20 0.35
SLC18A3 Q16572 1/20 0.34
TRPV6 Q9H1D0 1/20 0.34
L3MBTL3 Q96JM7 3/20 0.34
L3MBTL1 Q9Y468 3/20 0.34
RAB9A P51151 1/20 0.34
KCNK3 O14649 1/20 0.33
KCNK9 Q9NPC2 1/20 0.33
CDK1 P06493 1/20 0.33
CDK5 Q00535 1/20 0.33
KDM4A O75164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8586460 0.80 HTR1F (0.45) HTR1AHTR1DHTR1BHTR1FTMIGD3
SCHEMBL30909149 0.77 HTR1F (0.75) HTR1AHTR1DHTR1BHTR1F
SCHEMBL8386474 0.73 HTR1D (0.51) HTR1AHTR1DHTR1BHTR1F
SCHEMBL8721836 0.73 TMIGD3 (0.41) HTR1AHTR1DHTR1BHTR1FTMIGD3
SCHEMBL8383872 0.71 HTR1F (0.72) HTR1AHTR1DHTR1BHTR1F
SCHEMBL8386639 0.70 HTR1D (0.52) HTR1AHTR1DHTR1BHTR1F
SCHEMBL5309428 0.69 LRRK2 (0.42) HTR1AHTR1DHTR1BHTR1FRAB9A
SCHEMBL8381834 0.69 RAB9A (0.40) HTR1AHTR1DHTR1BHTR1FTMIGD3
SCHEMBL8387305 0.68 HTR1F (0.73) HTR1AHTR1DHTR1BHTR1F
SCHEMBL8586359 0.67 HTR1F (0.53) HTR1AHTR1DHTR1BHTR1FRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0875513-A1 Substituted heteroaromatic 5-HT 1F agonists ELI LILLY AND COMPANY (US) 1998-11-04 EP disclosed