SCHEMBL8725845

SCHEMBL8725845

CN(C)CCN(C(=O)c1ccc([NH])cc1)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2C P18825 1/20 0.51
MLYCD O95822 1/20 0.49
HPGD P15428 3/20 0.46
ALDH1A1 P00352 5/20 0.45
ADRB2 P07550 1/20 0.45
MEN1 O00255 4/20 0.45
KMT2A Q03164 4/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
TP53 P04637 1/20 0.44
EGFR P00533 1/20 0.43
ERBB2 P04626 1/20 0.43
PDK1 Q15118 1/20 0.43
OPRD1 P41143 1/20 0.43
NPC1 O15118 1/20 0.43
MAPT P10636 2/20 0.42
GLA P06280 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8725847 0.85 ADRA2C (0.55) ADRA2CMLYCDHPGDALDH1A1ADRB2
SCHEMBL7288882 0.80 ADRA2C (0.69) ADRA2CMLYCDHPGDALDH1A1ADRB2
SCHEMBL3152403 0.79 ADRA2C (0.55) ADRA2CHPGDALDH1A1MEN1KMT2A
SCHEMBL9325465 0.77 SMN1; SMN2 (0.56) ADRA2CALDH1A1MEN1KMT2ACYP3A4
SCHEMBL18457436 0.75 MEN1 (0.55) ALDH1A1MEN1KMT2ACYP3A4CYP2C9
SCHEMBL3162595 0.74 ALDH1A1 (0.73) ADRA2CALDH1A1MEN1KMT2ACYP3A4
SCHEMBL8446688 0.74 ALDH1A1 (0.60) ALDH1A1MEN1KMT2ASMN1; SMN2MAPT
SCHEMBL11572252 0.74 MEN1 (0.53) ADRA2CALDH1A1MEN1KMT2ACYP3A4
SCHEMBL9001626 0.74 ADRA2C (0.65) ADRA2CMLYCDHPGDALDH1A1ADRB2
SCHEMBL7290259 0.74 KDM4E (0.59) ADRA2CMLYCDALDH1A1ADRB2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832091-A1 C-4' MODIFIED ADENOSINE KINASE INHIBITORS GENSIA, INC. (US) 1998-04-01 EP disclosed
WO-1996040705-A1 C-4' MODIFIED ADENOSINE KINASE INHIBITORS GENSIA SICOR (US) 1996-12-19 WO disclosed