SCHEMBL8726244

SCHEMBL8726244

C[C@@H](C(=O)O)N(C)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.52
ADAMTS4 O75173 2/20 0.50
CYP1A2 P05177 1/20 0.47
GAA P10253 1/20 0.47
CYP2C9 P11712 1/20 0.47
PKM P14618 1/20 0.47
CYP2C19 P33261 1/20 0.47
FASN P49327 1/20 0.44
ALDH1A1 P00352 2/20 0.43
PDCD1 Q15116 1/20 0.43
CD274 Q9NZQ7 1/20 0.43
KDM4E B2RXH2 1/20 0.43
USP2 O75604 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
MAPT P10636 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
TAAR1 Q96RJ0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1997224 1.00 PTGS2 (0.52) PTGS2ADAMTS4CYP1A2GAACYP2C9
SCHEMBL755703 0.88 ALDH1A1 (0.43) PTGS2ADAMTS4ALDH1A1KDM4ESMN1; SMN2
SCHEMBL755702 0.88 ALDH1A1 (0.43) PTGS2ADAMTS4ALDH1A1KDM4ESMN1; SMN2
Hydrochloric Acid SCHEMBL8226909 0.86 ALDH1A1 (0.42) PTGS2ADAMTS4ALDH1A1KDM4ESMN1; SMN2
Hydrochloric Acid SCHEMBL32662705 0.86 ALDH1A1 (0.42) PTGS2ADAMTS4ALDH1A1KDM4ESMN1; SMN2
Hydrochloric Acid SCHEMBL8226911 0.86 ALDH1A1 (0.42) PTGS2ADAMTS4ALDH1A1KDM4ESMN1; SMN2
SCHEMBL10351875 0.84 PTGS2 (0.43) PTGS2ADAMTS4CYP1A2GAACYP2C9
SCHEMBL14969086 0.82 ADAMTS4 (0.59) PTGS2ADAMTS4CYP1A2GAACYP2C9
SCHEMBL8605929 0.81 ALDH1A1 (0.44) ALDH1A1SMN1; SMN2MAPTLMNA
SCHEMBL31370844 0.81 ALDH1A1 (0.44) ALDH1A1SMN1; SMN2MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780498-A PEPTIDE DERIVATIVES FOR CARDIOVASCULAR AND BRAIN DISORDERS CIBA-GEIGY JAPAN LIMITED (JP) 1998-07-14 US disclosed
EP-0728145-A1 ENDOTHELIN RECEPTOR ANTAGONISTS Ciba-Geigy Japan Limited (JP) 1996-08-28 EP disclosed
WO-1995012611-A1 ENDOTHELIN RECEPTOR ANTAGONISTS JAPAT LTD. (CH) 1995-05-11 WO disclosed