SCHEMBL8726261

SCHEMBL8726261

Cc1cc(C)cc(C(=O)N(C)[C@@H](Cc2ccc(O)cc2)C(=O)O)c1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 1/20 0.45
EDNRB P24530 10/20 0.41
EDNRA P25101 10/20 0.41
BACE1 P56817 1/20 0.38
BACE2 Q9Y5Z0 1/20 0.38
POLB P06746 1/20 0.37
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
FOLH1 Q04609 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8726257 1.00 SLC7A5 (0.45) SLC7A5EDNRBEDNRABACE1BACE2
SCHEMBL8721687 0.89 BACE1 (0.45) SLC7A5EDNRBEDNRABACE1BACE2
SCHEMBL8722642 0.89 BACE1 (0.45) SLC7A5EDNRBEDNRABACE1BACE2
SCHEMBL16907004 0.87 ALDH1A1 (0.50) EDNRBEDNRA
SCHEMBL7451078 0.87 ALDH1A1 (0.50) EDNRBEDNRA
SCHEMBL7451075 0.87 ALDH1A1 (0.50) EDNRBEDNRA
SCHEMBL8721883 0.86 ESR1 (0.47) EDNRBEDNRAESR1ESR2
SCHEMBL8721886 0.86 ESR1 (0.47) EDNRBEDNRAESR1ESR2
SCHEMBL8724800 0.86 LDHA (0.51) POLB
SCHEMBL8724804 0.86 LDHA (0.51) POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780498-A PEPTIDE DERIVATIVES FOR CARDIOVASCULAR AND BRAIN DISORDERS CIBA-GEIGY JAPAN LIMITED (JP) 1998-07-14 US disclosed
EP-0728145-A1 ENDOTHELIN RECEPTOR ANTAGONISTS Ciba-Geigy Japan Limited (JP) 1996-08-28 EP disclosed
WO-1995012611-A1 ENDOTHELIN RECEPTOR ANTAGONISTS JAPAT LTD. (CH) 1995-05-11 WO disclosed