SCHEMBL8724804

SCHEMBL8724804

COc1ccc(C[C@@H](C(=O)O)N(C)C(=O)c2cc(C)cc(C)c2)cc1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.51
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
TSPO P30536 1/20 0.45
PPARG P37231 2/20 0.42
PPARA Q07869 1/20 0.42
POLB P06746 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
TPH1 P17752 2/20 0.41
ACHE P22303 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8724800 1.00 LDHA (0.51) LDHAKMT2AMEN1TSPOPPARG
SCHEMBL8726261 0.86 SLC7A5 (0.45) POLB
SCHEMBL8726257 0.86 SLC7A5 (0.45) POLB
SCHEMBL8722642 0.85 BACE1 (0.45) KMT2AMEN1TSPOPOLBL3MBTL1
SCHEMBL8721687 0.85 BACE1 (0.45) KMT2AMEN1TSPOPOLBL3MBTL1
SCHEMBL8724369 0.85 TSPO (0.52) TSPOPPARGPPARA
SCHEMBL8724365 0.85 TSPO (0.52) TSPOPPARGPPARA
SCHEMBL7451075 0.84 ALDH1A1 (0.50) PPARGPPARA
SCHEMBL16907004 0.84 ALDH1A1 (0.50) PPARGPPARA
SCHEMBL7451078 0.84 ALDH1A1 (0.50) PPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780498-A PEPTIDE DERIVATIVES FOR CARDIOVASCULAR AND BRAIN DISORDERS CIBA-GEIGY JAPAN LIMITED (JP) 1998-07-14 US disclosed
EP-0728145-A1 ENDOTHELIN RECEPTOR ANTAGONISTS Ciba-Geigy Japan Limited (JP) 1996-08-28 EP disclosed
WO-1995012611-A1 ENDOTHELIN RECEPTOR ANTAGONISTS JAPAT LTD. (CH) 1995-05-11 WO disclosed