SCHEMBL8727112

SCHEMBL8727112

COc1ccc(Nc2[c]cccc2)cc1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 5/20 0.46
EGFR P00533 3/20 0.44
CLK1 P49759 1/20 0.44
STK10 O94804 1/20 0.44
SLK Q9H2G2 1/20 0.44
LCK P06239 1/20 0.43
ABCB1 P08183 2/20 0.43
ABCC1 P33527 2/20 0.43
FLT1 P17948 1/20 0.43
FLT4 P35916 1/20 0.43
KDR P35968 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
ALDH1A1 P00352 1/20 0.42
HTT P42858 1/20 0.42
FLT3 P36888 1/20 0.42
MAPT P10636 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8723583 0.84 APOBEC3A (0.52) EGFRLCKFLT1FLT4KDR
SCHEMBL6440705 0.78 RAB9A (0.55) SMN1; SMN2NPC1RAB9AALDH1A1HTT
SCHEMBL6986651 0.77 MEN1 (0.53) ABCG2EGFRCLK1ABCB1ABCC1
SCHEMBL8727116 0.76 EGFR (0.45) ABCG2EGFRCLK1LCKSMN1; SMN2
SCHEMBL8597483 0.75 MEN1 (0.62) ABCG2STK10SLKABCB1ABCC1
SCHEMBL27982530 0.75 KMT2A (0.53) EGFRNPC1ALDH1A1HTTMAPT
SCHEMBL4932459 0.75 MAPT (0.51) EGFRSMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL15389323 0.74 CCNK (0.43) EGFR
SCHEMBL8725290 0.74 POLB (0.41) EGFRALDH1A1HTTMAPTKDM4E
SCHEMBL6418064 0.72 HPGD (0.54) SMN1; SMN2NPC1RAB9AALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832091-A1 C-4' MODIFIED ADENOSINE KINASE INHIBITORS GENSIA, INC. (US) 1998-04-01 EP disclosed
WO-1996040705-A1 C-4' MODIFIED ADENOSINE KINASE INHIBITORS GENSIA SICOR (US) 1996-12-19 WO disclosed