SCHEMBL8728009

SCHEMBL8728009

CCOC(=O)c1ccc(Cc2ccc(NC(=O)OC(C)(C)C)cc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.60
NAMPT P43490 2/20 0.55
PDK1 Q15118 1/20 0.54
PDK2 Q15119 1/20 0.54
PDK3 Q15120 1/20 0.54
PDK4 Q16654 1/20 0.54
TSHR P16473 2/20 0.53
RAB9A P51151 8/20 0.53
NPC1 O15118 4/20 0.53
MAPT P10636 4/20 0.53
NPSR1 Q6W5P4 1/20 0.53
SMN1; SMN2 Q16637 5/20 0.52
MEN1 O00255 4/20 0.52
KMT2A Q03164 4/20 0.52
GAA P10253 2/20 0.52
CASP3 P42574 1/20 0.52
TRPV1 Q8NER1 1/20 0.52
SENP7 Q9BQF6 1/20 0.52
TP53 P04637 1/20 0.52
POLB P06746 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL273218 0.93 PDK1 (0.60) NAMPTPDK1PDK2PDK3PDK4
SCHEMBL132701 0.86 CYP17A1 (0.76) CYP17A1NAMPTTSHR
SCHEMBL14379115 0.83 CYP17A1 (0.68) CYP17A1NAMPTRAB9ANPC1SMN1; SMN2
SCHEMBL19945896 0.83 PDK1 (0.50) NAMPTPDK1PDK2PDK3PDK4
SCHEMBL10361607 0.81 CYP17A1 (0.61) CYP17A1NAMPTRAB9ASMN1; SMN2
SCHEMBL7143564 0.81 MEN1 (0.64) PDK1PDK2PDK3PDK4TSHR
SCHEMBL10249437 0.80 CYP17A1 (0.68) CYP17A1NAMPTRAB9ANPC1SMN1; SMN2
SCHEMBL10941324 0.80 NAMPT (0.69) NAMPTTSHRRAB9ANPC1MAPT
SCHEMBL3905352 0.80 HTT (0.59) NAMPTRAB9ANPC1MAPTSMN1; SMN2
SCHEMBL15709727 0.80 LMNA (0.62) CYP17A1TSHRMAPTSMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998035982-A1 COMPOUNDS FOR USE IN ADEPT ZENECA LIMITED (GB) 1998-08-20 WO disclosed