SCHEMBL8728811

SCHEMBL8728811

Cn1c(CC(=O)O)ccc1C(=O)c1ccc(-c2cccc(C(F)(F)F)c2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCL8 P10145 1/20 0.57
AKR1B1 P15121 1/20 0.57
PTGS1 P23219 1/20 0.57
PTGS2 P35354 1/20 0.57
GLO1 Q04760 1/20 0.57
HPGD P15428 1/20 0.46
S1PR5 Q9H228 1/20 0.43
SLC13A5 Q86YT5 1/20 0.43
CNR2 P34972 1/20 0.43
RXRA P19793 4/20 0.42
RXRB P28702 4/20 0.42
RXRG P48443 3/20 0.42
SRD5A2 P31213 1/20 0.42
KIF11 P52732 1/20 0.42
SLC6A7 Q99884 1/20 0.41
BACE1 P56817 1/20 0.41
SLC1A3 P43003 1/20 0.40
SLC1A2 P43004 1/20 0.40
SLC1A1 P43005 1/20 0.40
PLG P00747 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8726594 0.88 PTGS2 (0.65) CXCL8AKR1B1PTGS1PTGS2GLO1
SCHEMBL7678253 0.84 PTGS2 (0.70) CXCL8AKR1B1PTGS1PTGS2GLO1
SCHEMBL8458232 0.84 PTGS1 (0.74) CXCL8AKR1B1PTGS1PTGS2GLO1
SCHEMBL8728872 0.80 PTGS2 (0.70) CXCL8AKR1B1PTGS1PTGS2GLO1
SCHEMBL8732329 0.79 CXCL8 (0.56) CXCL8AKR1B1PTGS1PTGS2GLO1
SCHEMBL8729555 0.78 PTGS2 (0.72) CXCL8AKR1B1PTGS1PTGS2GLO1
SCHEMBL8729441 0.78 PTGS2 (0.91) CXCL8AKR1B1PTGS1PTGS2GLO1
SCHEMBL8728786 0.77 PTGS2 (0.60) CXCL8AKR1B1PTGS1PTGS2GLO1
Water SCHEMBL11371400 0.77 HPGD (0.57) CXCL8AKR1B1PTGS1PTGS2GLO1
SCHEMBL8733799 0.77 PTGS2 (0.70) CXCL8AKR1B1PTGS1PTGS2GLO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0783488-A4 FIVE MEMBERED HETEROCYCLIC COMPOUNDS ONO PHARMACEUTICAL CO (JP) 1998-01-07 EP claimed
EP-0783488-A1 FIVE MEMBERED HETEROCYCLIC COMPOUNDS ONO PHARMACEUTICAL CO., LTD. (JP) 1997-07-16 EP claimed
WO-1996010013-A1 FIVE MEMBERED HETEROCYCLIC COMPOUNDS ONO PHARMACEUTICAL CO., LTD. (JP) 1996-04-04 WO claimed