SCHEMBL8729117

SCHEMBL8729117

C[C@H](Cc1ccc(P(=O)(O)COc2ccccc2)cc1)NC(=O)OC(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.47
ADRB3 P13945 1/20 0.45
ACACB O00763 4/20 0.45
PTPN1 P18031 2/20 0.44
ATM Q13315 1/20 0.44
ITGB3 P05106 1/20 0.44
ITGA2B P08514 1/20 0.44
CTSS P25774 3/20 0.43
CTSK P43235 2/20 0.43
BCL2 P10415 1/20 0.43
CTSL P07711 1/20 0.43
CTSB P07858 1/20 0.43
PPARA Q07869 1/20 0.42
KLK5 Q9Y337 1/20 0.42
ACE P12821 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8729115 0.96 ADRB3 (0.49) HDAC8ADRB3ACACBPTPN1ATM
SCHEMBL8729106 0.96 ADRB3 (0.49) HDAC8ADRB3ACACBPTPN1ATM
SCHEMBL27460415 0.86 ACACB (0.45) HDAC8ACACBPTPN1ATMITGB3
SCHEMBL8732286 0.84 ACACB (0.49) HDAC8ADRB3ACACBPTPN1ITGB3
SCHEMBL8729119 0.84 ACACB (0.49) HDAC8ADRB3ACACBPTPN1ITGB3
SCHEMBL8729003 0.84 ACACB (0.49) HDAC8ADRB3ACACBPTPN1ITGB3
SCHEMBL3676166 0.80 NPC1 (0.63) ATMCTSSCTSKCTSLCTSB
SCHEMBL3676162 0.80 NPC1 (0.63) ATMCTSSCTSKCTSLCTSB
SCHEMBL12203694 0.80 NPC1 (0.63) ATMCTSSCTSKCTSLCTSB
SCHEMBL29401299 0.80 NPC1 (0.63) ATMCTSSCTSKCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5726165-A HYPOGLYCEMIC AGENTS; DIETETICS; GASTROINTESTINAL DISORDERS SMITHKLINE BEECHAM P.L.C. (GB) 1998-03-10 US disclosed