SCHEMBL8731622

SCHEMBL8731622

C=C/C(C)=C/C[C@@H]1[C@@]2(C)CCCC(C)(C)[C@@H]2C(O)C(O)[C@@]1(C)O

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.40
POLB P06746 1/20 0.40
CYP3A4 P08684 3/20 0.34
TP53 P04637 2/20 0.34
MAPK1 P28482 2/20 0.34
TRPC6 Q9Y210 1/20 0.34
ALOX15 P16050 1/20 0.34
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
ALDH1A1 P00352 1/20 0.32
TRPA1 O75762 1/20 0.32
CYP2C9 P11712 1/20 0.32
TSHR P16473 1/20 0.32
CYP2C19 P33261 1/20 0.32
LMNA P02545 1/20 0.31
UGT2B7 P16662 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29922526 1.00 MAPT (0.40) MAPTPOLBCYP3A4TP53MAPK1
SCHEMBL29551597 1.00 MAPT (0.40) MAPTPOLBCYP3A4TP53MAPK1
SCHEMBL30498603 0.83 MAPT (0.41) MAPTPOLBCYP3A4TP53MAPK1
SCHEMBL30498601 0.83 MAPT (0.38) MAPTPOLBCYP3A4TP53MAPK1
SCHEMBL8733660 0.80 TTL (0.39) MAPTPOLBCYP3A4TP53MAPK1
SCHEMBL8731624 0.77 MAPT (0.40) MAPTPOLBCYP3A4MEN1KMT2A
SCHEMBL8731628 0.71 ALDH1A1 (0.57) MAPTPOLBCYP3A4MEN1KMT2A
SCHEMBL18089046 0.71 ALDH1A1 (0.57) MAPTPOLBCYP3A4MEN1KMT2A
SCHEMBL9549996 0.71 ALDH1A1 (0.57) MAPTPOLBCYP3A4MEN1KMT2A
SCHEMBL15220009 0.71 ALDH1A1 (0.57) MAPTPOLBCYP3A4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5773005-A ENZYME INHIBITORS, ANTISECRETORY AGENTS AND ANTIANDROGENS KABUSHIKI KAISHA YAKURIGAKU CHUO KENKYUSHO (JP) 1998-06-30 US claimed
US-5773005-A ENZYME INHIBITORS, ANTISECRETORY AGENTS AND ANTIANDROGENS KABUSHIKI KAISHA YAKURIGAKU CHUO KENKYUSHO (JP) 1998-06-30 US disclosed
EP-0747048-A2 Diterpenes and flavonoids as 5-alpha-reductase inhibitors Kabushiki Kaisha Yakurigaku Chuo Kenkyusho (JP) 1996-12-11 EP disclosed