SCHEMBL8733222

SCHEMBL8733222

CCOC(=O)C(C(=O)OCC)C(=O)c1ccc(F)c(F)c1F

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.49
CES1 P23141 2/20 0.49
TSHR P16473 3/20 0.41
CA12 O43570 4/20 0.38
CA1 P00915 4/20 0.38
CA2 P00918 4/20 0.38
CA7 P43166 4/20 0.38
CA9 Q16790 4/20 0.38
CA14 Q9ULX7 4/20 0.38
NPSR1 Q6W5P4 3/20 0.37
HTT P42858 2/20 0.37
TP53 P04637 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
LMNA P02545 2/20 0.36
CYP1A2 P05177 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8731592 0.86 CES2 (0.36) CES2CES1TSHRNPSR1TDP1
SCHEMBL6779772 0.84 TSHR (0.37) TSHRCA12CA1CA2CA7
SCHEMBL8787463 0.84 CTSS (0.34) CES2CES1TSHRCA12CA1
SCHEMBL1958113 0.81 TSHR (0.57) CES2CES1TSHRCA12CA1
SCHEMBL9416413 0.79 CES2 (0.50) CES2CES1TSHRNPSR1TDP1
SCHEMBL9675530 0.76 MAPT (0.36) CES2CES1TSHRNPSR1HTT
SCHEMBL8165888 0.75 CES2 (0.58) CES2CES1ALDH1A1
SCHEMBL22261452 0.75 TSHR (0.53) CES2CES1TSHRCA12CA1
SCHEMBL29604715 0.75 TSHR (0.53) CES2CES1TSHRCA12CA1
SCHEMBL312535 0.74 CES2 (0.47) CES2CES1TSHRCA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0607824-B1 Method for the production of multiply halogenated benzotrichlorides and benzoyl chlorides as well as new multiply halogenated benzotrichlorides BAYER AG (DE) 1998-04-22 EP disclosed
EP-0607824-A2 Method for the production of multiply halogenated benzotrifluorides, benzotrichlorides and benzoyl chlorides as well as trihalobenzotrichlorides and -benzoyl chlorides BAYER AG (DE) 1994-07-27 EP disclosed
EP-0607825-A1 6-H-4-OXO-3-quinoline-carboxylic acids and their analogues as antibacterial agents BAYER AG (DE) 1994-07-27 EP disclosed