SCHEMBL8787463

SCHEMBL8787463

CCOC(=O)C(C(=O)OCC)C(=O)c1ccc(F)c(C(F)(F)F)c1F

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
NPSR1 Q6W5P4 2/20 0.34
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
POLB P06746 1/20 0.34
APP P05067 1/20 0.34
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
TSHR P16473 1/20 0.33
HPD P32754 1/20 0.32
HDAC4 P56524 2/20 0.32
HDAC6 Q9UBN7 2/20 0.32
HDAC3 O15379 1/20 0.32
HDAC1 Q13547 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8733222 0.84 CES2 (0.49) NPSR1CES2CES1MEN1LMNA
SCHEMBL8731592 0.80 CES2 (0.36) NPSR1CES2CES1POLBMEN1
SCHEMBL8926667 0.79 CES2 (0.39) CES2CES1TSHRKDM4ESMN1; SMN2
SCHEMBL9414350 0.78 APP (0.34) POLBAPPMEN1KMT2A
SCHEMBL28872705 0.74 HSP90AB1 (0.40) CES2CES1POLBMAPTTSHR
SCHEMBL22163772 0.74 LMNA (0.44) NPSR1POLBLMNACYP1A2MAPT
SCHEMBL8925622 0.74 NPSR1 (0.41) NPSR1CES2CES1POLBMEN1
SCHEMBL9416413 0.74 CES2 (0.50) NPSR1CES2CES1POLBMEN1
SCHEMBL8785757 0.73 NPSR1 (0.41) NPSR1CES2CES1POLBMEN1
SCHEMBL8925617 0.73 NPSR1 (0.41) NPSR1CES2CES1POLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0607826-B1 Fluoro-trifluoromethylbenzoic acid derivatives BAYER AG (DE) 1997-05-07 EP disclosed
EP-0607826-A1 Fluoro-Trifluoromethylbenzoic acid derivatives BAYER AG (DE) 1994-07-27 EP disclosed
EP-0607825-A1 6-H-4-OXO-3-quinoline-carboxylic acids and their analogues as antibacterial agents BAYER AG (DE) 1994-07-27 EP disclosed