SCHEMBL8733265

SCHEMBL8733265

Cn1c(CC(=O)O)ccc1C(=O)c1ccc(C#Cc2ccccc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.68
CXCL8 P10145 1/20 0.68
AKR1B1 P15121 1/20 0.68
PTGS1 P23219 1/20 0.68
GLO1 Q04760 1/20 0.68
HPGD P15428 1/20 0.51
FFAR1 O14842 5/20 0.49
GRM5 P41594 3/20 0.44
MMP2 P08253 3/20 0.43
MMP9 P14780 3/20 0.43
MMP12 P39900 3/20 0.43
MMP14 P50281 1/20 0.43
MMP15 P51511 1/20 0.43
MMP16 P51512 1/20 0.43
MMP26 Q9NRE1 1/20 0.43
ABCB11 O95342 1/20 0.40
FFAR4 Q5NUL3 1/20 0.40
PTGES O14684 1/20 0.38
ALOX5 P09917 1/20 0.38
HDAC10 Q969S8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8726561 0.87 PTGS2 (0.78) PTGS2CXCL8AKR1B1PTGS1GLO1
SCHEMBL2237360 0.87 PTGS2 (0.77) PTGS2CXCL8AKR1B1PTGS1GLO1
SCHEMBL7678784 0.85 PTGS2 (0.70) PTGS2CXCL8AKR1B1PTGS1GLO1
SCHEMBL8458232 0.85 PTGS1 (0.74) PTGS2CXCL8AKR1B1PTGS1GLO1
SCHEMBL8729681 0.82 PTGS2 (0.70) PTGS2CXCL8AKR1B1PTGS1GLO1
SCHEMBL8731019 0.82 PTGS2 (0.70) PTGS2CXCL8AKR1B1PTGS1GLO1
SCHEMBL8733815 0.82 CXCL8 (0.65) PTGS2CXCL8AKR1B1PTGS1GLO1
Tolmetin SCHEMBL11325188 0.81 PTGS2 (1.00) PTGS2CXCL8AKR1B1PTGS1GLO1
Tolmetin SCHEMBL3150 0.81 PTGS2 (1.00) PTGS2CXCL8AKR1B1PTGS1GLO1
SCHEMBL8729642 0.81 CXCL8 (0.68) PTGS2CXCL8AKR1B1PTGS1GLO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0783488-A4 FIVE MEMBERED HETEROCYCLIC COMPOUNDS ONO PHARMACEUTICAL CO (JP) 1998-01-07 EP claimed
EP-0783488-A1 FIVE MEMBERED HETEROCYCLIC COMPOUNDS ONO PHARMACEUTICAL CO., LTD. (JP) 1997-07-16 EP claimed
WO-1996010013-A1 FIVE MEMBERED HETEROCYCLIC COMPOUNDS ONO PHARMACEUTICAL CO., LTD. (JP) 1996-04-04 WO claimed