SCHEMBL8733807

SCHEMBL8733807

O=C1CC(Br)(Br)C(=O)c2c(F)cccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
CA7 P43166 2/20 0.50
CA9 Q16790 2/20 0.50
SRD5A1 P18405 2/20 0.36
AKR1A1 P14550 1/20 0.35
AKR1B1 P15121 1/20 0.35
DDB1 Q16531 1/20 0.34
CRBN Q96SW2 1/20 0.34
SLC6A9 P48067 1/20 0.33
PDK2 Q15119 1/20 0.33
TRPM8 Q7Z2W7 1/20 0.32
PGR P06401 1/20 0.31
ALDH1A1 P00352 1/20 0.31
KMT2A Q03164 2/20 0.30
MEN1 O00255 1/20 0.30
POLB P06746 1/20 0.30
WRN Q14191 1/20 0.30
MAPT P10636 1/20 0.30
RECQL P46063 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8599479 0.70 CA1 (0.46) CA1CA2CA7CA9SRD5A1
SCHEMBL14939549 0.70 MAPT (0.52) CA1CA2CA7CA9SRD5A1
SCHEMBL14939600 0.68 CA1 (0.57) CA1CA2CA7CA9AKR1A1
SCHEMBL22129686 0.67 CA1 (0.48) CA1CA2CA7CA9AKR1A1
SCHEMBL8665649 0.67 CA1 (1.00) CA1CA2CA7CA9AKR1A1
SCHEMBL31722364 0.64 SRD5A1 (0.47) CA1CA2CA7CA9SRD5A1
SCHEMBL5866470 0.64 CA1 (0.52) CA1CA2CA7CA9AKR1A1
SCHEMBL13487412 0.64 CA1 (0.52) CA1CA2CA7CA9AKR1A1
SCHEMBL10716838 0.64 MAOA (0.52) CA1CA2CA7CA9AKR1A1
SCHEMBL14939579 0.62 SRD5A1 (0.36) CA1CA2CA7CA9SRD5A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0876356-A1 USE OF TRICYCLIC 1,4-DIHYDRO-1,4-DIOXO-1H-NAPHTHALENE DERIVATIVES, RESULTING NOVEL COMPOUNDS AND THERAPEUTICAL USE THEREOF LABORATOIRE INNOTHERA Société Anonyme (FR) 1998-11-11 EP disclosed
WO-1997021684-A1 USE OF TRICYCLIC 1,4-DIHYDRO-1,4-DIOXO-1H-NAPHTHALENE DERIVATIVES, RESULTING NOVEL COMPOUNDS AND THERAPEUTICAL USE THEREOF LABORATOIRE INNOTHERA, SOCIETE ANONYME (FR) 1997-06-19 WO disclosed