SCHEMBL8734706

SCHEMBL8734706

O=C(O)Cc1ccc2c(c1)CC(CNS(=O)(=O)c1cccs1)C2

nearest known ligand 0.82

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 7/20 0.82
ALDH1A1 P00352 4/20 0.50
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
APOB P04114 1/20 0.49
MTTP P55157 1/20 0.49
HPGD P15428 2/20 0.48
TP53 P04637 2/20 0.47
TSHR P16473 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8731670 0.85 TBXA2R (0.82) TBXA2RMEN1KMT2A
SCHEMBL8734189 0.82 TBXA2R (0.64) TBXA2R
SCHEMBL8734661 0.80 TBXA2R (0.70) TBXA2R
SCHEMBL8730165 0.80 TBXA2R (0.70) TBXA2R
SCHEMBL8730048 0.80 TBXA2R (0.70) TBXA2RMEN1KMT2A
SCHEMBL8734691 0.80 TBXA2R (0.70) TBXA2RALDH1A1MEN1KMT2A
SCHEMBL8733779 0.80 TBXA2R (0.70) TBXA2R
SCHEMBL5673556 0.80 TBXA2R (0.85) TBXA2R
SCHEMBL8728396 0.79 TBXA2R (0.63) TBXA2RALDH1A1
SCHEMBL8734677 0.79 TBXA2R (0.84) TBXA2RALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750524-A ADMINISTERING AN SULFAMIDE SUBSTITUTED INDAN DERIVATIVE ZERIA PHARMACEUTICAL CO., LTD. (JP) 1998-05-12 US disclosed
EP-0773019-A1 HYPERLIPEMIA REMEDY ZERIA PHARMACEUTICAL CO., LTD. (JP) 1997-05-14 EP disclosed
EP-0589037-B1 INDIAN DERIVATIVE AND THROMBOXANE ANTAGONIST CONTAINING THE SAME ZERIA PHARM CO LTD (JP) 1996-05-29 EP disclosed
US-5409956-A A sulfonylaminoalkylindan carboxylic acid or ester for treating thrombosis, vasospasm or asthma ZERIA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0589037-A1 INDIAN DERIVATIVE AND THROMBOXANE ANTAGONIST CONTAINING THE SAME ZERIA PHARMACEUTICAL CO., LTD. (JP) 1994-03-30 EP disclosed