SCHEMBL8735820

SCHEMBL8735820

Cc1cc2cc(F)ccc2nc1-c1ccc(-c2ccccc2)cc1

nearest known ligand 0.65

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.65
DHODH Q02127 14/20 0.57
PDK1 Q15118 1/20 0.50
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
MAPK14 Q16539 1/20 0.46
MBNL1 Q9NR56 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
DHFR P00374 1/20 0.45
ALKBH5 Q6P6C2 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28536199 0.97 PDE10A (0.69) PDE10ADHODHPDK1KDM4EALDH1A1
SCHEMBL8735048 0.87 DHODH (0.62) PDE10ADHODHPDK1ALDH1A1
SCHEMBL8733061 0.86 DHODH (0.53) PDE10ADHODHPDK1MAPK14MBNL1
SCHEMBL8732571 0.85 DHODH (0.62) PDE10ADHODHMBNL1DHFRALKBH5
SCHEMBL29942008 0.85 DHODH (0.62) PDE10ADHODHMBNL1DHFRALKBH5
SCHEMBL28085639 0.83 PDE10A (0.74) PDE10APDK1MAPK14MBNL1TDP1
SCHEMBL14341086 0.83 PDE10A (0.93) PDE10ADHODHPDK1KDM4EALDH1A1
SCHEMBL12970097 0.80 PDK1 (0.47) PDE10ADHODHPDK1KDM4EMAPK14
SCHEMBL12970115 0.80 PDK1 (0.45) PDE10ADHODHPDK1KDM4EMAPK14
SCHEMBL28529940 0.80 PDE10A (0.73) PDE10ADHODHKDM4EALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0537191-B1 TREATMENT OF ORGAN TRANSPLANTATION REJECTION DU PONT MERCK PHARMA (US) 1998-04-29 EP claimed
EP-0339485-B1 4-QUINOLINE CARBOXYLIC ACID DERIVATIVES USEFUL AS IMMUNOSUPPRESSIVE AGENTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1993-03-31 EP claimed