SCHEMBL8738130

SCHEMBL8738130

CC(C)c1cccc(-c2cccnc2N)c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.63
ABL1 P00519 1/20 0.44
SRC P12931 1/20 0.44
MKNK1 Q9BUB5 1/20 0.43
MKNK2 Q9HBH9 1/20 0.43
KDR P35968 1/20 0.41
RXRA P19793 2/20 0.40
RXRB P28702 1/20 0.40
RXRG P48443 1/20 0.40
TGFBR1 P36897 1/20 0.39
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39
PDE4A P27815 2/20 0.38
PDE4B Q07343 2/20 0.38
PDE4C Q08493 2/20 0.38
PDE4D Q08499 2/20 0.38
USP7 Q93009 1/20 0.38
ADK P55263 1/20 0.38
FYN P06241 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15340847 0.82 MKNK1 (0.43) MAP4K4ABL1SRCMKNK1MKNK2
SCHEMBL624495 0.81 MKNK1 (0.54) MAP4K4MKNK1MKNK2TGFBR1NOS3
SCHEMBL15496384 0.79 PDE4B (0.50) PDE4APDE4BPDE4CPDE4DBRD4
SCHEMBL14881894 0.79 RXRA (0.52) KDRRXRARXRBRXRGNR4A2
SCHEMBL15340953 0.78 ALOX5AP (0.47) KDRPDE4APDE4BPDE4CPDE4D
SCHEMBL13524662 0.78 ACVR1 (0.50) FYNCREBBP
SCHEMBL4582784 0.78 MAP4K4 (0.69) MAP4K4ABL1MKNK1MKNK2KDR
SCHEMBL9177215 0.77 RXRA (0.50) KDRRXRARXRBRXRGBRD4
SCHEMBL398059 0.76 ALDH1A1 (0.52) ABL1SRCKDRRXRARXRB
SCHEMBL18188070 0.76 MAP4K4 (0.71) MAP4K4MKNK1MKNK2NOS3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012068589-A2 MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF CONSTELLATION PHARMACEUTICALS (US) 2012-05-24 WO disclosed