SCHEMBL8738231

SCHEMBL8738231

O=C(N[C@H]1CCN(Cc2ccccc2)C1)c1ccc(Oc2ccccc2)cc1

nearest known ligand 0.87

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 13/20 0.77
DRD4 P21917 13/20 0.77
SLC2A1 P11166 1/20 0.74
MCHR1 Q99705 1/20 0.69
HTR2A P28223 1/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8738579 1.00 DRD2 (0.77) DRD2DRD4SLC2A1MCHR1HTR2A
SCHEMBL7218171 0.93 TMEM97 (0.74) DRD2DRD4MCHR1
SCHEMBL7694199 0.89 DRD2 (0.85) DRD2DRD4MCHR1HTR2A
SCHEMBL7694198 0.89 DRD2 (0.85) DRD2DRD4MCHR1HTR2A
SCHEMBL11555632 0.87 DRD2 (0.82) DRD2DRD4MCHR1HTR2A
SCHEMBL8706290 0.87 DRD2 (1.00) DRD2DRD4MCHR1HTR2A
SCHEMBL8707354 0.87 DRD2 (1.00) DRD2DRD4MCHR1HTR2A
SCHEMBL2900269 0.86 TMEM97 (0.86) DRD2DRD4MCHR1HTR2A
SCHEMBL8236258 0.86 TMEM97 (0.86) DRD2DRD4MCHR1HTR2A
SCHEMBL8706273 0.84 DRD2 (0.89) DRD2DRD4HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012068589-A2 MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF CONSTELLATION PHARMACEUTICALS (US) 2012-05-24 WO disclosed