SCHEMBL8739096

SCHEMBL8739096

C=C(Cl)CC1(C(=O)N[C@@H](Cc2ccc(-c3ccccc3)cc2)/C(N)=N/N=N)CCCC1

nearest known ligand 0.47

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 17/20 0.44
ITGA4 P13612 17/20 0.44
MMP1 P03956 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3698356 0.81 MMP1 (0.66) ITGB1ITGA4MMP1
SCHEMBL3698358 0.81 MMP1 (0.66) ITGB1ITGA4MMP1
SCHEMBL3701146 0.80 MMP1 (0.48) ITGB1ITGA4MMP1
SCHEMBL3701143 0.80 MMP1 (0.48) ITGB1ITGA4MMP1
SCHEMBL7539221 0.74 PSMB1 (0.48) ITGB1ITGA4MMP1
SCHEMBL7540140 0.74 ITGB1 (0.67) ITGB1ITGA4
SCHEMBL3709738 0.74 ITGB1 (0.67) ITGB1ITGA4
SCHEMBL3709737 0.74 ITGB1 (0.67) ITGB1ITGA4
SCHEMBL8739536 0.74 HDAC1 (0.52) ITGB1ITGA4MMP1
SCHEMBL16214799 0.72 ITGB1 (0.39) ITGB1ITGA4MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012065953-A1 SUBSTITUTED CARBAMOYLCYCLOALKYL ACETIC ACID DERIVATIVES AS NEP INHIBITORS NOVARTIS AG (CH) 2012-05-24 WO disclosed