SCHEMBL8739201

SCHEMBL8739201

CC1(C)CC(NC(=O)c2ccc(Cn3cnc4ccccc43)cc2)CC(C)(C)N1

nearest known ligand 0.61

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.61
HDAC6 Q9UBN7 1/20 0.61
EZH2 Q15910 8/20 0.58
HRH3 Q9Y5N1 4/20 0.49
IDO1 P14902 4/20 0.49
LMNA P02545 1/20 0.48
CYP11B1 P15538 1/20 0.48
CYP11B2 P19099 1/20 0.48
HTT P42858 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9302839 0.82 HDAC1 (0.67) HDAC1HDAC6HRH3IDO1LMNA
SCHEMBL8738652 0.78 MEN1 (0.57) EZH2HTTMEN1KMT2A
SCHEMBL12850040 0.77 HDAC6 (1.00) HDAC1HDAC6IDO1LMNACYP11B1
Tert-Butyl Formate SCHEMBL27786473 0.76 HDAC1 (0.53) HDAC1HDAC6HRH3IDO1LMNA
SCHEMBL8738670 0.76 EZH2 (0.74) EZH2MEN1KMT2A
SCHEMBL6120593 0.76 EZH2 (0.74) EZH2MEN1KMT2A
SCHEMBL3725969 0.76 HDAC1 (0.55) HDAC1HDAC6HRH3LMNAMEN1
SCHEMBL28787442 0.76 HDAC1 (0.52) HDAC1HDAC6HRH3IDO1LMNA
SCHEMBL8738903 0.75 EZH2 (0.53) EZH2MEN1KMT2A
SCHEMBL169747 0.75 EZH2 (0.80) EZH2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012068589-A2 MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF CONSTELLATION PHARMACEUTICALS (US) 2012-05-24 WO disclosed