SCHEMBL28787442

SCHEMBL28787442

CC(C)(C)C(=O)OC1C[C@@H](NC(=O)c2ccc(Cn3cnc4ccccc43)cc2)CN1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
HRH3 Q9Y5N1 7/20 0.43
IDO1 P14902 5/20 0.43
CYP11B1 P15538 4/20 0.41
CYP11B2 P19099 4/20 0.41
HTT P42858 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
LMNA P02545 2/20 0.41
TSHR P16473 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MAPK1 P28482 1/20 0.40
TNF P01375 1/20 0.39
MGLL Q99685 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28787440 0.81 CRHR1 (0.40) HDAC6SMN1; SMN2TSHR
SCHEMBL27808373 0.81 CRHR1 (0.40) HDAC6SMN1; SMN2TSHR
SCHEMBL27808326 0.79 HDAC1 (0.49) HDAC1HDAC6HRH3HTTSMN1; SMN2
SCHEMBL27808501 0.79 HDAC1 (0.49) HDAC1HDAC6HRH3HTTSMN1; SMN2
SCHEMBL27808277 0.77 KHK (0.49) HRH3CYP11B1CYP11B2MAPK1
SCHEMBL27786338 0.77 GCG (0.44) HRH3
SCHEMBL9302839 0.76 HDAC1 (0.67) HDAC1HDAC6HRH3IDO1CYP11B1
SCHEMBL8739201 0.76 HDAC1 (0.61) HDAC1HDAC6HRH3IDO1CYP11B1
Tert-Butyl Formate SCHEMBL27786473 0.75 HDAC1 (0.53) HDAC1HDAC6HRH3IDO1CYP11B1
SCHEMBL3725969 0.75 HDAC1 (0.55) HDAC1HDAC6HRH3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101778838-A Azacyclylbenzamide derivatives as histamine-3 antagonists WYETH CORP 2010-07-14 CN disclosed