SCHEMBL9302839

SCHEMBL9302839

O=C(NC1CCCCC1)c1ccc(Cn2cnc3ccccc32)cc1

nearest known ligand 0.67

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.67
HDAC6 Q9UBN7 1/20 0.67
HRH3 Q9Y5N1 6/20 0.56
IDO1 P14902 3/20 0.53
RXFP1 Q9HBX9 1/20 0.53
GAA P10253 1/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
KMT2A Q03164 1/20 0.53
TP53 P04637 1/20 0.52
LMNA P02545 1/20 0.52
CYP11B1 P15538 2/20 0.51
CYP11B2 P19099 2/20 0.51
TNF P01375 1/20 0.51
MAPK1 P28482 1/20 0.51
HTT P42858 1/20 0.51
KDM4E B2RXH2 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9303119 0.88 FAAH (0.60) HDAC1HDAC6HRH3IDO1KMT2A
SCHEMBL8739201 0.82 HDAC1 (0.61) HDAC1HDAC6HRH3IDO1SMN1; SMN2
SCHEMBL3725969 0.82 HDAC1 (0.55) HDAC1HDAC6HRH3KMT2ATP53
SCHEMBL12850040 0.81 HDAC6 (1.00) HDAC1HDAC6IDO1SMN1; SMN2LMNA
Tert-Butyl Formate SCHEMBL27786473 0.80 HDAC1 (0.53) HDAC1HDAC6HRH3IDO1SMN1; SMN2
SCHEMBL4937775 0.79 HTT (0.51) HDAC1HDAC6HRH3IDO1SMN1; SMN2
SCHEMBL4943222 0.78 USP30 (0.56) HDAC1HDAC6HRH3
SCHEMBL4943219 0.78 USP30 (0.56) HDAC1HDAC6HRH3
SCHEMBL9303184 0.78 CYP11B1 (0.51) HDAC1HDAC6HRH3GAASMN1; SMN2
SCHEMBL4937782 0.76 LMNA (0.54) HDAC1HDAC6HRH3IDO1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5314880-A Platelet activating factor antagonist BRITISH BIO-TECHNOLOGY LIMITED (GB) 1994-05-24 US disclosed
EP-0468971-A1 NOVEL BENZIMIDAZOLE DERIVATIVES BRITISH BIO-TECHNOLOGY LIMITED (GB) 1992-02-05 EP disclosed
WO-1990009997-A1 NOVEL BENZIMIDAZOLE DERIVATIVES BRITISH BIO-TECHNOLOGY LIMITED (GB) 1990-09-07 WO disclosed