SCHEMBL8740581

SCHEMBL8740581

CCCC(I)c1ccc(OC)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
TAS1R3 Q7RTX0 1/20 0.44
TAS1R1 Q7RTX1 1/20 0.44
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C19 P33261 1/20 0.43
ALDH1A1 P00352 3/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MIF P14174 1/20 0.42
MMP1 P03956 1/20 0.41
MMP13 P45452 1/20 0.41
CYP17A1 P05093 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8741660 0.83 MIF (0.49) CA12CA1CA2CA7CA9
SCHEMBL1198451 0.79 ALDH1A1 (0.49) CA12CA1CA2CA7CA9
SCHEMBL4742927 0.79 CYP17A1 (0.51) CA12CA1CA2CA7CA9
SCHEMBL23343772 0.78 ABCB11 (0.49) CA12CA1CA2CA7CA9
SCHEMBL28343944 0.78 ALDH1A1 (0.50) CA12CA1CA2CA7CA9
SCHEMBL10052129 0.78 ALDH1A1 (0.50) CA12CA1CA2CA7CA9
SCHEMBL8276044 0.77 CHRNA7 (0.38) CA12CA2CA9CYP2C19ALDH1A1
SCHEMBL3645373 0.77 ALDH1A1 (0.40) CA12CA1CA2CA7CA9
SCHEMBL20011556 0.77 KDM4E (0.39) CA12CA2ALDH1A1MMP1MMP13
SCHEMBL5488204 0.76 AOC3 (0.58) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733044-A4 COMPOUNDS SMITHKLINE BEECHAM CORP (US) 1997-03-05 EP disclosed
EP-0733044-A1 COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1996-09-25 EP disclosed
EP-0649412-A4 PHARMACEUTICAL PYRIDINE COMPOUNDS. SMITHKLINE BEECHAM CORP (US) 1995-07-05 EP disclosed
WO-1995015950-A1 COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1995-06-15 WO disclosed
EP-0649412-A1 PHARMACEUTICAL PYRIDINE COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1995-04-26 EP disclosed
WO-1994000437-A1 PHARMACEUTICAL PYRIDINE COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1994-01-06 WO disclosed