SCHEMBL8740658

SCHEMBL8740658

O=P(O)(O)C(O)c1cccc(Oc2ccccc2)c1

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PGK1 P00558 2/20 0.65
PGK2 P07205 2/20 0.65
PTGS1 P23219 1/20 0.55
MEN1 O00255 1/20 0.50
CYP2D6 P10635 1/20 0.50
KMT2A Q03164 1/20 0.50
ALOX5 P09917 1/20 0.48
MMP2 P08253 1/20 0.47
MMP8 P22894 1/20 0.47
MMP14 P50281 1/20 0.47
CA9 Q16790 1/20 0.47
CA14 Q9ULX7 1/20 0.47
AKR1C3 P42330 1/20 0.46
HDAC8 Q9BY41 1/20 0.45
SRC P12931 1/20 0.44
FDFT1 P37268 1/20 0.43
ACP3 P15309 1/20 0.42
NPY5R Q15761 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9007810 0.89 PGK1 (0.59) PGK1PGK2PTGS1MEN1CYP2D6
SCHEMBL9007806 0.88 PGK1 (0.57) PGK1PGK2PTGS1MEN1CYP2D6
SCHEMBL9007812 0.88 PGK1 (0.57) PGK1PGK2PTGS1MEN1CYP2D6
SCHEMBL9007805 0.88 PGK1 (0.57) PGK1PGK2PTGS1MEN1CYP2D6
SCHEMBL8740626 0.86 PGK1 (0.59) PGK1PGK2PTGS1CYP2D6ACP3
SCHEMBL9007814 0.83 PGK1 (0.56) PGK1PGK2PTGS1MMP8MMP14
SCHEMBL11214240 0.83 PTGS1 (0.55) PGK1PGK2PTGS1MEN1CYP2D6
SCHEMBL9007809 0.82 PGK1 (0.54) PGK1PGK2PTGS1ACP3
SCHEMBL11046075 0.79 POLB (0.70) PTGS1MEN1CYP2D6KMT2AALOX5
SCHEMBL11388011 0.79 PTGS1 (0.57) PTGS1MEN1CYP2D6KMT2AALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0746323-A4 1997-01-22 EP disclosed
EP-0746323-A1 INHIBITORS OF PHOSPHOINOSITIDE-SPECIFIC PHOSPHOLIPASE C MERCK & CO. INC. (US) 1996-12-11 EP disclosed
US-5519163-A A-HYDROXYPHOSPHONATE COMPOUNDS MERCK & CO., INC. (US) 1996-05-21 US disclosed
WO-1995010286-A1 INHIBITORS OF PHOSPHOINOSITIDE-SPECIFIC PHOSPHOLIPASE C MERCK & CO., INC. (US) 1995-04-20 WO disclosed
US-4471118-A Preparation of aldehydes by heating an α-hydroxyphosphonic acid ester BAYER AKTIENGESELLSCHAFT (DE) 1984-09-11 US disclosed