SCHEMBL8743531

SCHEMBL8743531

O=CC(F)(F)COCc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.50
KDM4E B2RXH2 1/20 0.47
POLB P06746 1/20 0.47
ALDH1A1 P00352 3/20 0.45
NPSR1 Q6W5P4 1/20 0.40
CES1 P23141 1/20 0.40
AR P10275 1/20 0.40
TACR1 P25103 1/20 0.40
PTPN2 P17706 1/20 0.39
PTPN1 P18031 1/20 0.39
PTPN6 P29350 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A3 Q01959 1/20 0.39
KMT2A Q03164 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CA1 P00915 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8157722 0.78 ALDH1A1 (0.61) TSHRKDM4EPOLBALDH1A1NPSR1
SCHEMBL4889465 0.78 TSHR (0.50) TSHRKDM4EPOLBALDH1A1AR
SCHEMBL2398930 0.78 TSHR (0.50) TSHRKDM4EPOLBALDH1A1CA1
SCHEMBL23273064 0.77 TSHR (0.45) TSHRKDM4EPOLBALDH1A1NPSR1
SCHEMBL8743631 0.76 TSHR (0.44) TSHRKDM4EPOLBALDH1A1TACR1
SCHEMBL23273063 0.76 TSHR (0.44) TSHRKDM4EPOLBALDH1A1NPSR1
SCHEMBL9521927 0.75 TSHR (0.47) TSHRKDM4EPOLBALDH1A1AR
SCHEMBL18526730 0.75 KDM4E (0.53) TSHRKDM4EPOLBALDH1A1AR
SCHEMBL28991495 0.75 TSHR (0.42) TSHRKDM4EPOLBALDH1A1NPSR1
Potassium Ion SCHEMBL29823215 0.75 TSHR (0.42) TSHRKDM4EPOLBALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0335770-B1 Novel fluorophosphonate nucleotide derivatives MERRELL PHARMA INC (US) 1997-01-15 EP disclosed
EP-0339161-A1 Novel fluorophosphonate nucleotide derivatives MERRELL DOW PHARMACEUTICALS INC. (US) 1989-11-02 EP disclosed
EP-0335770-A2 Novel fluorophosphonate nucleotide derivatives MERRELL PHARMACEUTICALS INC. (US) 1989-10-04 EP disclosed