SCHEMBL8744222

SCHEMBL8744222

CCCC[Si](C)(C)[C@]1(n2cc(C)c(=O)[nH]c2=O)C[C@H](O)[C@@H](CO)O1

nearest known ligand 0.41

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TK2 O00142 5/20 0.41
TK1 P04183 5/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3300455 0.87 RNASE1 (0.37) TK2TK1
SCHEMBL27561054 0.86 TK1 (0.43) TK2TK1
SCHEMBL20379162 0.86 TYMP (0.41) TK2TK1
SCHEMBL16267748 0.85 SLC28A1 (0.38) TK2TK1
SCHEMBL8145394 0.82 TK1 (0.42) TK2TK1
SCHEMBL28238519 0.82 TK1 (0.40) TK2TK1
SCHEMBL5163085 0.80 TK2 (0.43) TK2TK1
SCHEMBL29587983 0.79 TK2 (0.44) TK2TK1
SCHEMBL29364921 0.78 TK1 (0.45) TK1
SCHEMBL9396543 0.78 RNASE1 (0.39) TK2TK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3356381-A1 DESIGN AND SYNTHESIS OF NOVEL DISULFIDE LINKER BASED NUCLEOTIDES AS REVERSIBLE TERMINATORS FOR DNA SEQUENCING BY SYNTHESIS The Trustees of Columbia University in the City of New York (US) 2018-08-08 EP disclosed
EP-0753002-A1 MODIFIED OLIGONUCLEOTIDES AND INTERMEDIATES USEFUL IN NUCLEIC ACID THERAPEUTICS AMGEN INC. (US) 1997-01-15 EP disclosed
EP-0707591-A1 METHYLPHOSPHONIC ACID ESTER, PROCESS FOR PREPARING THE SAME AND ITS USE HOECHST AKTIENGESELLSCHAFT (DE) 1996-04-24 EP disclosed
WO-1995026972-A1 MODIFIED OLIGONUCLEOTIDES AND INTERMEDIATES USEFUL IN NUCLEIC ACID THERAPEUTICS AMGEN INC. (US) 1995-10-12 WO disclosed
WO-1994022883-A1 BACKBONE MODIFIED OLIGONUCLEOTIDES AND THEIR PREPARATION ISIS PHARMACEUTICALS, INC. (US) 1994-10-13 WO disclosed
WO-1994022893-A1 OLIGONUCLEOSIDE LINKAGES CONTAINING ADJACENT NITROGEN ATOMS ISIS PHARMACEUTICALS, INC. (US) 1994-10-13 WO disclosed
WO-1994022454-A1 OLIGONUCLEOSIDE LINKAGES CONTAINING ADJACENT OXYGEN AND NITROGEN ATOMS ISIS PHARMACEUTICALS, INC. (US) 1994-10-13 WO disclosed
EP-0064796-B1 PHOSPHORYLATING AGENT AND PROCESS FOR THE PHOSPHORYLATION OF ORGANIC HYDROXYL COMPOUNDS UNILEVER N.V. (NL) 1985-05-15 EP disclosed