SCHEMBL8744762

SCHEMBL8744762

CCOC(=O)[C@H](Cc1ccccc1)NC(=O)Cc1c(Cl)cccc1Cl

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.56
POLB P06746 1/20 0.51
ALDH1A1 P00352 2/20 0.50
PTGS2 P35354 1/20 0.50
TACR1 P25103 1/20 0.50
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
NOS3 P29474 1/20 0.49
NOS1 P29475 1/20 0.49
NOS2 P35228 1/20 0.49
GAA P10253 1/20 0.48
RAB9A P51151 1/20 0.48
PRSS1 P07477 1/20 0.48
PRSS2 P07478 1/20 0.48
PRSS3 P35030 1/20 0.48
MMP8 P22894 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11559927 0.87 TP53 (0.60) TP53POLBALDH1A1TACR1MEN1
SCHEMBL8744724 0.85 PRSS1 (0.57) PRSS1PRSS2PRSS3
SCHEMBL8744720 0.85 PRSS1 (0.57) PRSS1PRSS2PRSS3
SCHEMBL8744805 0.84 TACR1 (0.57) TP53POLBALDH1A1TACR1MEN1
SCHEMBL9594563 0.84 TACR1 (0.57) TP53POLBALDH1A1TACR1MEN1
SCHEMBL9594765 0.84 PPID (0.46) TP53POLBALDH1A1KMT2ANOS3
SCHEMBL8744783 0.84 PPID (0.46) TP53POLBALDH1A1KMT2ANOS3
SCHEMBL9488184 0.83 TP53 (0.59) TP53POLBALDH1A1PTGS2TACR1
SCHEMBL9488182 0.83 TP53 (0.59) TP53POLBALDH1A1PTGS2TACR1
SCHEMBL9487298 0.83 TP53 (0.61) TP53POLBALDH1A1TACR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0456063-B1 1-H-3-aryl-pyrrolidin-2,4-dion-derivatives BAYER AG (DE) 1997-01-22 EP disclosed
EP-0456063-A2 1-H-3-aryl-pyrrolidin-2,4-dion-derivatives BAYER AG (DE) 1991-11-13 EP disclosed