SCHEMBL8744783

SCHEMBL8744783

CCOC(=O)[C@H](CC(C)C)NC(=O)Cc1c(Cl)cccc1Cl

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PPID Q08752 1/20 0.46
NOS3 P29474 2/20 0.46
NOS1 P29475 2/20 0.46
NOS2 P35228 2/20 0.46
ALDH1A1 P00352 4/20 0.43
MAPT P10636 3/20 0.43
HTT P42858 1/20 0.43
KMT2A Q03164 1/20 0.43
PTPN11 Q06124 1/20 0.42
SLC22A12 Q96S37 1/20 0.42
ANPEP P15144 1/20 0.41
POLB P06746 2/20 0.41
HPGD P15428 1/20 0.41
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
LMNA P02545 2/20 0.41
TP53 P04637 2/20 0.40
THRB P10828 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9594765 1.00 PPID (0.46) PPIDNOS3NOS1NOS2ALDH1A1
SCHEMBL9594560 0.84 KMT2A (0.47) ALDH1A1MAPTHTTKMT2ASLC22A12
SCHEMBL8744777 0.84 KMT2A (0.47) ALDH1A1MAPTHTTKMT2ASLC22A12
SCHEMBL8744789 0.84 GRN (0.56) ALDH1A1KMT2ASLC22A12LMNATP53
SCHEMBL8744785 0.84 GRN (0.56) ALDH1A1KMT2ASLC22A12LMNATP53
SCHEMBL8744762 0.84 TP53 (0.56) NOS3NOS1NOS2ALDH1A1KMT2A
SCHEMBL8744727 0.82 KMT2A (0.44) ALDH1A1MAPTHTTKMT2ASLC22A12
SCHEMBL9594623 0.82 KMT2A (0.44) ALDH1A1MAPTHTTKMT2ASLC22A12
SCHEMBL4426485 0.81 NOS3 (0.51) NOS3NOS1NOS2ALDH1A1TAS1R3
SCHEMBL9595460 0.81 LMNA (0.51) PPIDALDH1A1POLBHPGDTAS1R3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0456063-B1 1-H-3-aryl-pyrrolidin-2,4-dion-derivatives BAYER AG (DE) 1997-01-22 EP disclosed
US-5258527-A Insecticidal, acaricidal and herbicidal 1-H-3-aryl-pyrrolidine-2,4-dione derivatives BAYER AKTIENGESELLSCHAFT (DE) 1993-11-02 US disclosed
EP-0456063-A2 1-H-3-aryl-pyrrolidin-2,4-dion-derivatives BAYER AG (DE) 1991-11-13 EP disclosed