SCHEMBL8744765

SCHEMBL8744765

O=C(O)CNC(=O)Cc1c(Cl)cccc1Cl

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.63
SMN1; SMN2 Q16637 1/20 0.56
KMT2A Q03164 3/20 0.56
POLB P06746 1/20 0.51
SHMT1 P34896 2/20 0.51
SHMT2 P34897 2/20 0.51
P2RX7 Q99572 6/20 0.49
RECQL P46063 1/20 0.48
SIGMAR1 Q99720 1/20 0.46
ATM Q13315 1/20 0.46
ADRA2A P08913 2/20 0.45
MEN1 O00255 1/20 0.45
LMNA P02545 1/20 0.45
CYP3A4 P08684 1/20 0.45
HTR1A P08908 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
ADRA2B P18089 1/20 0.45
ADRA2C P18825 1/20 0.45
MAOA P21397 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12836854 0.81 AKR1B1 (0.45) AKR1B1SMN1; SMN2KMT2APOLBSHMT1
SCHEMBL109215 0.78 AKR1B1 (1.00) AKR1B1SMN1; SMN2KMT2ARECQLADRA2A
SCHEMBL8744812 0.78 SMN1; SMN2 (0.63) SMN1; SMN2KMT2AP2RX7ATMMEN1
SCHEMBL13485815 0.77 KMT2A (0.62) AKR1B1SMN1; SMN2KMT2ARECQLSIGMAR1
Hydrochloric Acid SCHEMBL1374156 0.77 AKR1B1 (0.95) AKR1B1SMN1; SMN2KMT2ARECQLADRA2A
SCHEMBL9364446 0.77 AKR1B1 (0.95) AKR1B1SMN1; SMN2KMT2ARECQLADRA2A
SCHEMBL13329784 0.76 KMT2A (0.62) AKR1B1SMN1; SMN2KMT2AP2RX7RECQL
SCHEMBL9527443 0.76 KMT2A (0.61) AKR1B1SMN1; SMN2KMT2AP2RX7RECQL
SCHEMBL25279561 0.75 RECQL (0.68) AKR1B1SMN1; SMN2KMT2ARECQLATM
SCHEMBL2854479 0.75 KMT2A (0.61) SMN1; SMN2KMT2APOLBP2RX7MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0456063-B1 1-H-3-aryl-pyrrolidin-2,4-dion-derivatives BAYER AG (DE) 1997-01-22 EP disclosed
US-5258527-A Insecticidal, acaricidal and herbicidal 1-H-3-aryl-pyrrolidine-2,4-dione derivatives BAYER AKTIENGESELLSCHAFT (DE) 1993-11-02 US disclosed
EP-0456063-A2 1-H-3-aryl-pyrrolidin-2,4-dion-derivatives BAYER AG (DE) 1991-11-13 EP disclosed