SCHEMBL8744812

SCHEMBL8744812

CCOC(=O)CNC(=O)Cc1c(Cl)cccc1Cl

nearest known ligand 0.63

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.63
HTT P42858 1/20 0.58
MAPK1 P28482 1/20 0.49
NLRP3 Q96P20 1/20 0.49
P2RX7 Q99572 3/20 0.48
KMT2A Q03164 2/20 0.48
GAA P10253 2/20 0.47
PPID Q08752 1/20 0.47
MEN1 O00255 1/20 0.45
ATM Q13315 1/20 0.45
ALDH1A1 P00352 1/20 0.45
RAB9A P51151 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1429298 0.82 AKR1B1 (0.55) SMN1; SMN2HTTMAPK1NLRP3KMT2A
Ammonia Solution, Strong SCHEMBL27532390 0.81 AKR1B1 (0.53) SMN1; SMN2HTTMAPK1NLRP3KMT2A
SCHEMBL11305630 0.80 NLRP3 (0.52) SMN1; SMN2HTTMAPK1NLRP3KMT2A
SCHEMBL4003642 0.80 HTT (0.55) SMN1; SMN2HTTNLRP3KMT2APPID
SCHEMBL18754170 0.79 HTT (0.60) SMN1; SMN2HTTNLRP3PPIDALDH1A1
SCHEMBL8744765 0.78 AKR1B1 (0.63) SMN1; SMN2MAPK1P2RX7KMT2AMEN1
SCHEMBL30385493 0.77 PPID (0.66) KMT2AGAAPPIDMEN1ALDH1A1
SCHEMBL8744815 0.76 GAA (0.56) HTTP2RX7KMT2AGAAMEN1
SCHEMBL9594560 0.75 KMT2A (0.47) SMN1; SMN2HTTMAPK1NLRP3P2RX7
SCHEMBL8744777 0.75 KMT2A (0.47) SMN1; SMN2HTTMAPK1NLRP3P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0456063-B1 1-H-3-aryl-pyrrolidin-2,4-dion-derivatives BAYER AG (DE) 1997-01-22 EP disclosed
US-5258527-A Insecticidal, acaricidal and herbicidal 1-H-3-aryl-pyrrolidine-2,4-dione derivatives BAYER AKTIENGESELLSCHAFT (DE) 1993-11-02 US disclosed
EP-0456063-A2 1-H-3-aryl-pyrrolidin-2,4-dion-derivatives BAYER AG (DE) 1991-11-13 EP disclosed