SCHEMBL8744831

SCHEMBL8744831

CCOC(=O)[C@H](Cc1ccc(OC)cc1)NC(=O)Cc1c(C)cc(C)cc1C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
L3MBTL1 Q9Y468 1/20 0.46
EPHX2 P34913 1/20 0.46
ITGB1 P05556 1/20 0.45
ITGA4 P13612 1/20 0.45
TACR1 P25103 2/20 0.44
HTT P42858 1/20 0.43
LDHA P00338 1/20 0.43
GLA P06280 1/20 0.43
KMT2A Q03164 1/20 0.43
TP53 P04637 1/20 0.43
PSMB5 P28074 1/20 0.42
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC8 Q9BY41 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9594665 1.00 ALDH1A1 (0.50) ALDH1A1L3MBTL1EPHX2ITGB1ITGA4
SCHEMBL8744826 0.89 ITGB1 (0.54) ALDH1A1L3MBTL1ITGB1ITGA4LDHA
SCHEMBL8744821 0.89 ITGB1 (0.54) ALDH1A1L3MBTL1ITGB1ITGA4LDHA
SCHEMBL8744805 0.88 TACR1 (0.57) ALDH1A1L3MBTL1TACR1KMT2ATP53
SCHEMBL9594563 0.88 TACR1 (0.57) ALDH1A1L3MBTL1TACR1KMT2ATP53
SCHEMBL11674845 0.82 ACACB (0.54) ALDH1A1EPHX2TACR1LDHAGLA
SCHEMBL14370512 0.82 ACACB (0.54) ALDH1A1EPHX2TACR1LDHAGLA
SCHEMBL4403600 0.79 ALDH1A1 (0.55) ALDH1A1GLAKMT2AHDAC3HDAC4
SCHEMBL26148921 0.79 GAA (0.54) ALDH1A1EPHX2GAARAB9A
SCHEMBL28356496 0.79 HDAC8 (0.60) ALDH1A1KMT2AHDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0456063-B1 1-H-3-aryl-pyrrolidin-2,4-dion-derivatives BAYER AG (DE) 1997-01-22 EP disclosed
US-5258527-A Insecticidal, acaricidal and herbicidal 1-H-3-aryl-pyrrolidine-2,4-dione derivatives BAYER AKTIENGESELLSCHAFT (DE) 1993-11-02 US disclosed